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Target
Cathepsin G
Ligand
BDBM50249353
Substrate
n/a
Meas. Tech.
ChEMBL_499484 (CHEMBL1021976)
IC50
433200±n/a nM
Citation
 Martins, FT; Assis, DM; Dos Santos, MH; Camps, I; Veloso, MP; Juliano, MA; Alves, LC; Doriguetto, AC Natural polyprenylated benzophenones inhibiting cysteine and serine proteases. Eur J Med Chem 44:1230-9 (2009) [PubMed]  Article 
Target
Name:
Cathepsin G
Synonyms:
CATG_HUMAN | CG | CTSG
Type:
PROTEIN
Mol. Mass.:
28860.08
Organism:
Homo sapiens (Human)
Description:
ChEMBL_1469016
Residue:
255
Sequence:
MQPLLLLLAFLLPTGAEAGEIIGGRESRPHSRPYMAYLQIQSPAGQSRCGGFLVREDFVLTAAHCWGSNINVTLGAHNIQRRENTQQHITARRAIRHPQYNQRTIQNDIMLLQLSRRVRRNRNVNPVALPRAQEGLRPGTLCTVAGWGRVSMRRGTDTLREVQLRVQRDRQCLRIFGSYDPRRQICVGDRRERKAAFKGDSGGPLLCNNVAHGIVSYGKSSGVPPEVFTRVSSFLPWIRTTMRSFKLLDQMETPL
  
Inhibitor
Name:
BDBM50249353
Synonyms:
1,1,3-trihydroxybenzophenone | 2,2',4-trihydroxybenzophenone | CHEMBL470701 | Polyhydroxy benzophenone, 13
Type:
Small organic molecule
Emp. Form.:
C13H10O4
Mol. Mass.:
230.2161
SMILES:
Oc1ccc(C(=O)c2ccccc2O)c(O)c1
Structure:
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