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Target
Transcriptional activator protein LuxR
Ligand
BDBM50350710
Substrate
n/a
Meas. Tech.
ChEMBL_762767 (CHEMBL1816069)
IC50
770±n/a nM
Citation
McInnis, CE; Blackwell, HE Thiolactone modulators of quorum sensing revealed through library design and screening. Bioorg Med Chem 19:4820-8 (2011) [PubMed] Article
More Info.:
Target
Name:
Transcriptional activator protein LuxR
Synonyms:
LUXR_ALIFS | luxR
Type:
PROTEIN
Mol. Mass.:
28563.86
Organism:
Vibrio fischeri
Description:
ChEMBL_831639
Residue:
250
Sequence:
MKNINADDTYRIINKIKACRSNNDINQCLSDMTKMVHCEYYLLAIIYPHSMVKSDISILDNYPKKWRQYYDDANLIKYDPIVDYSNSNHSPINWNIFENNAVNKKSPNVIKEAKTSGLITGFSFPIHTANNGFGMLSFAHSEKDNYIDSLFLHACMNIPLIVPSLVDNYRKINIANNKSNNDLTKREKECLAWACEGKSSWDISKILGCSERTVTFHLTNAQMKLNTTNRCQSISKAILTGAIDCPYFKN