Reaction Details Report a problem with these data
Target
Non-secretory ribonuclease
Ligand
BDBM50402338
Substrate
n/a
Meas. Tech.
ChEMBL_885938 (CHEMBL2215700)
Ki
180±n/a nM
Citation
Parmenopoulou, V; Chatzileontiadou, DS; Manta, S; Bougiatioti, S; Maragozidis, P; Gkaragkouni, DN; Kaffesaki, E; Kantsadi, AL; Skamnaki, VT; Zographos, SE; Zounpoulakis, P; Balatsos, NA; Komiotis, D; Leonidas, DD Triazole pyrimidine nucleosides as inhibitors of Ribonuclease A. Synthesis, biochemical, and structural evaluation. Bioorg Med Chem 20:7184-93 (2012) [PubMed] Article
More Info.:
Target
Name:
Non-secretory ribonuclease
Synonyms:
EDN | Eosinophil-derived neurotoxin (EDN) | Non-secretory ribonuclease | RNAS2_HUMAN | RNASE2 | RNAse 2 | RNS2
Type:
Protein
Mol. Mass.:
18364.09
Organism:
Homo sapiens (Human)
Description:
n/a
Residue:
161
Sequence:
MVPKLFTSQICLLLLLGLLAVEGSLHVKPPQFTWAQWFETQHINMTSQQCTNAMQVINNYQRRCKNQNTFLLTTFANVVNVCGNPNMTCPSNKTRKNCHHSGSQVPLIHCNLTTPSPQNISNCRYAQTPANMFYIVACDNRDQRRDPPQYPVVPVHLDRII