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Target
Beta-2 adrenergic receptor
Ligand
BDBM50405021
Substrate
n/a
Meas. Tech.
ChEMBL_37999 (CHEMBL651633)
Kd
30902.95±n/a nM
Citation
 Bouzoubaa, M; Leclerc, G; Decker, N; Schwartz, J; Andermann, G Synthesis and beta-adrenergic blocking activity of new aliphatic and alicyclic oxime ethers. J Med Chem 27:1291-4 (1984) [PubMed]  Article 
Target
Name:
Beta-2 adrenergic receptor
Synonyms:
ADRB2_CAVPO | Adrb2 | adrenergic Beta2
Type:
Enzyme Catalytic Domain
Mol. Mass.:
46993.24
Organism:
GUINEA PIG
Description:
adrenergic Beta2 ADRB2 GUINEA PIG::Q8K4Z4
Residue:
418
Sequence:
MGHLGNGSDFLLAPNASHAPDHNVTRERDEAWVVGMAIVMSLIVLAIVFGNVLVITAIAKFERLQTVTNYFITSLACADLVMGLAVVPFGASHILMNMWTFGNFWCEFWTSIDVLCVTASIETLCVIAVDRYFAITSPFKYQSLLTKNKARVVILMVWVVSGLTSFLPIQMHWYRATHKDAINCYAEETCCDFFTNQAYAIASSIVSFYLPLVVMVFVYSRVFQVAKKQLQKIDRSEGRFHTQNLSQVEQDGRSGHGLRRSSKFYLKEHKALKTLGIIMGTFTLCWLPFFIVNIVHVIQDNLIPKEVYILLNWVGYVNSAFNPLIYCRSPDFRIAFQELLCLRRSALKAYGNDCSSNSNGKTDYTGEPNVCHQGQEKERELLCEDPPGTEDLVSCPGTVPSDSIDSQGRNYSTNDSLL
  
Inhibitor
Name:
BDBM50405021
Synonyms:
CHEMBL26607
Type:
Small organic molecule
Emp. Form.:
C14H27NO2
Mol. Mass.:
241.3697
SMILES:
CC(C)(C)NCC(O)COC(C1CC1)C1CC1
Structure:
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