Reaction Details Report a problem with these data
Target
Emopamil-binding protein-like
Ligand
BDBM50334158
Substrate
n/a
Meas. Tech.
ChEMBL_936215 (CHEMBL2320419)
Ki
1400±n/a nM
Citation
 Wang, X; Li, Y; Deuther-Conrad, W; Xie, F; Chen, X; Cui, MC; Zhang, XJ; Zhang, JM; Steinbach, J; Brust, P; Liu, BL; Jia, HM Synthesis and biological evaluation of¹8F labeled fluoro-oligo-ethoxylated 4-benzylpiperazine derivatives for sigma-1 receptor imaging. Bioorg Med Chem 21:215-22 (2012) [PubMed]  Article 
Target
Name:
Emopamil-binding protein-like
Synonyms:
EBPL | EBPL_HUMAN | EBRP | ERP | Emopamil-binding-related protein
Type:
PROTEIN
Mol. Mass.:
23203.44
Organism:
Homo sapiens (Human)
Description:
ChEMBL_936215
Residue:
206
Sequence:
MGAEWELGAEAGGSLLLCAALLAAGCALGLRLGRGQGAADRGALIWLCYDALVHFALEGPFVYLSLVGNVANSDGLIASLWKEYGKADARWVYFDPTIVSVEILTVALDGSLALFLIYAIVKEKYYRHFLQITLCVCELYGCWMTFLPEWLTRSPNLNTSNWLYCWLYLFFFNGVWVLIPGLLLWQSWLELKKMHQKETSSVKKFQ
  
Inhibitor
Name:
BDBM50334158
Synonyms:
1'-benzyl-3-(2-fluoroethyl)-3H-spiro[[2]benzofuran-1,4'-piperidine | CHEMBL1645202 | CHEMBL2314421
Type:
Small organic molecule
Emp. Form.:
C21H24FNO
Mol. Mass.:
325.4198
SMILES:
FCCC1OC2(CCN(Cc3ccccc3)CC2)c2ccccc12
Structure:
Search PDB for entries with ligand similarity: