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Target
Emopamil-binding protein-like
Ligand
BDBM50424041
Substrate
n/a
Meas. Tech.
ChEMBL_936215 (CHEMBL2320419)
Ki
1.7±n/a nM
Citation
 Wang, X; Li, Y; Deuther-Conrad, W; Xie, F; Chen, X; Cui, MC; Zhang, XJ; Zhang, JM; Steinbach, J; Brust, P; Liu, BL; Jia, HM Synthesis and biological evaluation of¹8F labeled fluoro-oligo-ethoxylated 4-benzylpiperazine derivatives for sigma-1 receptor imaging. Bioorg Med Chem 21:215-22 (2012) [PubMed]  Article 
Target
Name:
Emopamil-binding protein-like
Synonyms:
EBPL | EBPL_HUMAN | EBRP | ERP | Emopamil-binding-related protein
Type:
PROTEIN
Mol. Mass.:
23203.44
Organism:
Homo sapiens (Human)
Description:
ChEMBL_936215
Residue:
206
Sequence:
MGAEWELGAEAGGSLLLCAALLAAGCALGLRLGRGQGAADRGALIWLCYDALVHFALEGPFVYLSLVGNVANSDGLIASLWKEYGKADARWVYFDPTIVSVEILTVALDGSLALFLIYAIVKEKYYRHFLQITLCVCELYGCWMTFLPEWLTRSPNLNTSNWLYCWLYLFFFNGVWVLIPGLLLWQSWLELKKMHQKETSSVKKFQ
  
Inhibitor
Name:
BDBM50424041
Synonyms:
CHEMBL2314420
Type:
Small organic molecule
Emp. Form.:
C22H30N2O3
Mol. Mass.:
370.4852
SMILES:
COc1ccc(CCN2CCN(CCCc3ccccc3)CC2)cc1OO
Structure:
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