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Target
N-arachidonyl glycine receptor
Ligand
BDBM50434876
Substrate
n/a
Meas. Tech.
ChEMBL_963378 (CHEMBL2388875)
IC50
>10000±n/a nM
Citation
 Rempel, V; Volz, N; Gläser, F; Nieger, M; Bräse, S; Müller, CE Antagonists for the orphan G-protein-coupled receptor GPR55 based on a coumarin scaffold. J Med Chem 56:4798-810 (2013) [PubMed]  Article 
Target
Name:
N-arachidonyl glycine receptor
Synonyms:
G-protein coupled receptor 18 | GPCRW | GPR18 | GPR18_HUMAN | NAGly receptor
Type:
PROTEIN
Mol. Mass.:
38150.44
Organism:
Homo sapiens (Human)
Description:
ChEMBL_107601
Residue:
331
Sequence:
MITLNNQDQPVPFNSSHPDEYKIAALVFYSCIFIIGLFVNITALWVFSCTTKKRTTVTIYMMNVALVDLIFIMTLPFRMFYYAKDEWPFGEYFCQILGALTVFYPSIALWLLAFISADRYMAIVQPKYAKELKNTCKAVLACVGVWIMTLTTTTPLLLLYKDPDKDSTPATCLKISDIIYLKAVNVLNLTRLTFFFLIPLFIMIGCYLVIIHNLLHGRTSKLKPKVKEKSIRIIITLLVQVLVCFMPFHICFAFLMLGTGENSYNPWGAFTTFLMNLSTCLDVILYYIVSKQFQARVISVMLYRNYLRSMRRKSFRSGSLRSLSNINSEML
  
Inhibitor
Name:
BDBM50434876
Synonyms:
CHEMBL2387539
Type:
Small organic molecule
Emp. Form.:
C20H20O3
Mol. Mass.:
308.371
SMILES:
Cc1ccccc1Cc1cc2c(C)c(O)c(C)c(C)c2oc1=O
Structure:
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