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Target
Dual specificity protein kinase CLK2
Ligand
BDBM50347750
Substrate
n/a
Meas. Tech.
ChEMBL_1280769 (CHEMBL3097753)
IC50
320±n/a nM
Citation
Burgy, G; Tahtouh, T; Durieu, E; Foll-Josselin, B; Limanton, E; Meijer, L; Carreaux, F; Bazureau, JP Chemical synthesis and biological validation of immobilized protein kinase inhibitory Leucettines. Eur J Med Chem 62:728-37 (2013) [PubMed] Article
More Info.:
Target
Name:
Dual specificity protein kinase CLK2
Synonyms:
CDC-like kinase 2 | CLK2_MOUSE | Clk2
Type:
PROTEIN
Mol. Mass.:
60021.57
Organism:
Mus musculus
Description:
ChEMBL_1502246
Residue:
499
Sequence:
MPHPRRYHSSERGSRGSYHEHYQSRKHKRRRSRSWSSSSDRTRRRRREDSYHVRSRSSYDDHSSDRRLYDRRYCGSYRRNDYSRDRGEAYYDTDFRQSYEYHRENSSYRSQRSSRRKHRRRRRRSRTFSRSSSHSSRRAKSVEDDAEGHLIYHVGDWLQERYEIVSTLGEGTFGRVVQCVDHRRGGTQVALKIIKNVEKYKEAARLEINVLEKINEKDPDNKNLCVQMFDWFDYHGHMCISFELLGLSTFDFLKDNNYLPYPIHQVRHMAFQLCQAVKFLHDNKLTHTDLKPENILFVNSDYELTYNLEKKRDERSVKSTAVRVVDFGSATFDHEHHSTIVSTRHYRAPEVILELGWSQPCDVWSIGCIIFEYYVGFTLFQTHDNREHLAMMERILGPVPSRMIRKTRKQKYFYRGRLDWDENTSAGRYVRENCKPLRRYLTSEAEDHHQLFDLIENMLEYEPAKRLTLGEALQHPFFACLRTEPPNTKLWDSSRDISR