Reaction Details Report a problem with these data
Target
Free fatty acid receptor 3
Ligand
BDBM50107305
Substrate
n/a
Meas. Tech.
ChEMBL_1508992 (CHEMBL3602372)
EC50
>10000±n/a nM
Citation
 Zahanich, I; Kondratov, I; Naumchyk, V; Kheylik, Y; Platonov, M; Zozulya, S; Krasavin, M Phenoxymethyl 1,3-oxazoles and 1,2,4-oxadiazoles as potent and selective agonists of free fatty acid receptor 1 (GPR40). Bioorg Med Chem Lett 25:3105-11 (2015) [PubMed]  Article 
Target
Name:
Free fatty acid receptor 3
Synonyms:
FFAR3 | FFAR3_HUMAN | GPR41
Type:
PROTEIN
Mol. Mass.:
38655.15
Organism:
Homo sapiens (Human)
Description:
ChEMBL_1508992
Residue:
346
Sequence:
MDTGPDQSYFSGNHWFVFSVYLLTFLVGLPLNLLALVVFVGKLQRRPVAVDVLLLNLTASDLLLLLFLPFRMVEAANGMHWPLPFILCPLSGFIFFTTIYLTALFLAAVSIERFLSVAHPLWYKTRPRLGQAGLVSVACWLLASAHCSVVYVIEFSGDISHSQGTNGTCYLEFRKDQLAILLPVRLEMAVVLFVVPLIITSYCYSRLVWILGRGGSHRRQRRVAGLLAATLLNFLVCFGPYNVSHVVGYICGESPAWRIYVTLLSTLNSCVDPFVYYFSSSGFQADFHELLRRLCGLWGQWQQESSMELKEQKGGEEQRADRPAERKTSEHSQGCGTGGQVACAES
  
Inhibitor
Name:
BDBM50107305
Synonyms:
CHEMBL3601001
Type:
Small organic molecule
Emp. Form.:
C19H18N2O4
Mol. Mass.:
338.3572
SMILES:
Cc1ccc(cc1)-c1noc(COc2ccc(CCC(O)=O)cc2)n1
Structure:
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