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Target
Cereblon isoform 4
Ligand
BDBM50146598
Substrate
n/a
Meas. Tech.
ChEMBL_1555511 (CHEMBL3768093)
Kd
3300±n/a nM
Citation
 Boichenko, I; Deiss, S; Bär, K; Hartmann, MD; Hernandez Alvarez, B A FRET-Based Assay for the Identification and Characterization of Cereblon Ligands. J Med Chem 59:770-4 (2016) [PubMed]  Article 
Target
Name:
Cereblon isoform 4
Synonyms:
Cereblon isoform 4
Type:
PROTEIN
Mol. Mass.:
13620.40
Organism:
Magnetospirillum gryphiswaldense
Description:
ChEMBL_116733
Residue:
124
Sequence:
MPLDAGGQNSTQMVLAPGASIFRCRQCGQTISRRDWLLPMGGDHEHVVFNPAGMIFRVWCFSLAQGLRLIGAPSGEFSWFKGYDWTIALCGQCGSHLGWHYEGGSQPQTFFGLIKDRLAEGPAD
  
Inhibitor
Name:
BDBM50146598
Synonyms:
CHEMBL3764647
Type:
Small organic molecule
Emp. Form.:
C14H16N4O3
Mol. Mass.:
288.3018
SMILES:
CNc1ccccc1C(=O)NCCn1ccc(=O)[nH]c1=O
Structure:
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