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Target
Chromobox protein homolog 3
Ligand
BDBM50194259
Substrate
n/a
Meas. Tech.
ChEMBL_1616639 (CHEMBL3858708)
Kd
>100000±n/a nM
Citation
Stuckey, JI; Simpson, C; Norris-Drouin, JL; Cholensky, SH; Lee, J; Pasca, R; Cheng, N; Dickson, BM; Pearce, KH; Frye, SV; James, LI Structure-Activity Relationships and Kinetic Studies of Peptidic Antagonists of CBX Chromodomains. J Med Chem 59:8913-8923 (2016) [PubMed] Article
More Info.:
Target
Name:
Chromobox protein homolog 3
Synonyms:
CBX3 | CBX3_HUMAN | Chromobox protein homolog 3 | HECH | HP1 gamma | Heterochromatin protein 1 homolog gamma | Modifier 2 protein
Type:
PROTEIN
Mol. Mass.:
20806.65
Organism:
Homo sapiens (Human)
Description:
ChEMBL_116825
Residue:
183
Sequence:
MASNKTTLQKMGKKQNGKSKKVEEAEPEEFVVEKVLDRRVVNGKVEYFLKWKGFTDADNTWEPEENLDCPELIEAFLNSQKAGKEKDGTKRKSLSDSESDDSKSKKKRDAADKPRGFARGLDPERIIGATDSSGELMFLMKWKDSDEADLVLAKEANMKCPQIVIAFYEERLTWHSCPEDEAQ