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Target
5-hydroxytryptamine receptor 4
Ligand
BDBM82505
Substrate
n/a
Ki
0.1±n/a nM
Comments
PDSP_1672
Citation
 Van den Wyngaert, I; Gommeren, W; Verhasselt, P; Jurzak, M; Leysen, J; Luyten, W; Bender, E Cloning and expression of a human serotonin 5-HT4 receptor cDNA. J Neurochem 69:1810-9 (1997) [PubMed]  Article 
Target
Name:
5-hydroxytryptamine receptor 4
Synonyms:
5-HT-4 | 5-HT4 | 5-HT4S | 5-HT4a | 5-HT4b | 5-HT4c | 5-HT4d | 5-HT4hb | 5-hydroxytryptamine receptor 4 | 5-hydroxytryptamine receptor 4 (5-HT4) | 5HT4R_HUMAN | HTR4 | Serotonin (5-HT) receptor | Serotonin (5-HT3) receptor | Serotonin 4 (5-HT4) receptor | Serotonin Receptor 4
Type:
Enzyme
Mol. Mass.:
43767.54
Organism:
Homo sapiens (Human)
Description:
Q13639
Residue:
388
Sequence:
MDKLDANVSSEEGFGSVEKVVLLTFLSTVILMAILGNLLVMVAVCWDRQLRKIKTNYFIVSLAFADLLVSVLVMPFGAIELVQDIWIYGEVFCLVRTSLDVLLTTASIFHLCCISLDRYYAICCQPLVYRNKMTPLRIALMLGGCWVIPTFISFLPIMQGWNNIGIIDLIEKRKFNQNSNSTYCVFMVNKPYAITCSVVAFYIPFLLMVLAYYRIYVTAKEHAHQIQMLQRAGASSESRPQSADQHSTHRMRTETKAAKTLCIIMGCFCLCWAPFFVTNIVDPFIDYTVPGQVWTAFLWLGYINSGLNPFLYAFLNKSFRRAFLIILCCDDERYRRPSILGQTVPCSTTTINGSTHVLRDAVECGGQWESQCHPPATSPLVAAQPSDT
  
Inhibitor
Name:
BDBM82505
Synonyms:
CAS_121881 | NSC_121881 | SB204070
Type:
Small organic molecule
Emp. Form.:
C19H27ClN2O4
Mol. Mass.:
382.882
SMILES:
CCCCN1CCC(COC(=O)c2cc(Cl)c(N)c3OCCOc23)CC1
Structure:
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