Reaction Details
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Report a problem with these dataTarget
Melatonin receptor type 1B
Ligand
BDBM85239
Substrate
n/a
Ki
0.55±n/a nM
Comments
PDSP_178
Citation
Sugden, D; Pickering, H; Teh, MT; Garratt, PJ Melatonin receptor pharmacology: toward subtype specificity. Biol Cell 89:531-7 (1997) [PubMed] Article More Info.:
Target
Name:
Melatonin receptor type 1B
Synonyms:
MEL-1B-R | MTR1B_CHICK | Melatonin | Melatonin receptor | Melatonin receptor type 1B
Type:
Enzyme Catalytic Domain
Mol. Mass.:
33012.73
Organism:
Chick
Description:
Melatonin 0 Chick::P51050
Residue:
289
Sequence:
GNAFVVSLALADLVVALYPYPLVLLAIFHNGWTLGEMHCKVSGFVMGLSVIGSIFNITAIAINRYCYICHSFAYDKVYSCWNTMLYVSLIWVLTVIATVPNFFVGSLKYDPRIYSCTFVQTASSYYTIAVVVIHFIVPITVVSFCYLRIWVLVLQVRRRVKSETKPRLKPSDFRNFLTMFVVFVIFAFCWAPLNFIGLAVAINPSEMAPKVPEWLFIISYFMAYFNSCLNAIIYGLLNQNFRNEYKRILMSLWMPRLFFQDTSKGGTDGQKSKPSPALNNNDQMKTDTL
Inhibitor
Name:
BDBM85239
Synonyms:
5-MeOT-N-propionyl
Type:
Small organic molecule
Emp. Form.:
C17H23N3O2
Mol. Mass.:
301.3834
SMILES:
CCC(=O)NCCc1ccc2[nH]cc(CCNC(C)=O)c2c1
Structure:
