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Target
Aromatase [1-48]
Ligand
BDBM85250
Substrate
n/a
Meas. Tech.
Biological Assay
IC50
200±n/a nM
Citation
 Pouget, C; Yahiaoui, S; Fagnere, C; Habrioux, G; Chulia, AJ Synthesis and biological evaluation of 4-imidazolylflavans as nonsteroidal aromatase inhibitors. Bioorg Chem 32:494-503 (2004) [PubMed]  Article 
Target
Name:
Aromatase [1-48]
Synonyms:
Aromatase cytochrome P450 | CP19A_HUMAN | CYP19A1 | ARO1 | CYAR | CYP19
Type:
Protein
Mol. Mass.:
5299.77
Organism:
Human
Description:
Q16449
Residue:
48
Sequence:
MVLEMLNPIHYNITSIVPEAMPAATMPVLLLTGLFLLVWNYEGTSSIP
  
Inhibitor
Name:
BDBM85250
Synonyms:
2,4-Trans-4'-chloro-4-imidazolyl-7-methoxyflavan, 3b
Type:
Small organic molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
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