Reaction Details Report a problem with these data
Target
Alpha-1A adrenergic receptor
Ligand
BDBM81444
Substrate
n/a
Ki
15.85±n/a nM
Comments
PDSP_1955
Citation
Wikberg-Matsson, A; Wikberg, JE; Uhlén, S Characterization of alpha1-adrenoceptor subtypes in the pig. Eur J Pharmacol 347:301-9 (1998) [PubMed] Article
More Info.:
Target
Name:
Alpha-1A adrenergic receptor
Synonyms:
ADA1A_CAVPO | ADRA1A | adrenergic Alpha1A
Type:
Enzyme Catalytic Domain
Mol. Mass.:
51603.72
Organism:
PIG
Description:
adrenergic Alpha1A ADRA1A PIG::Q9WU25
Residue:
466
Sequence:
MVFLSGNASDSSNCTQPPAPVNIPKAILLGVILGVLILFGVPGNILVILSVACHRHLHSVTHYYIVNLAVADLLLTSTVLPFSAIFEILGYWAFGRVFCNIWAAVDVLCCTASIMSLCIISIDRYIGVSYPLRYPTIVTQRRGLRALLCLWALSLVISIGPLFGWRQPAPQDETICQINEDPSYVLFSALGSFYVPLAIILVMYCRVYVVAKRESRGLTSGLKTDKSDSEQVTLRIHRKNAPLGGSGVASSKNKTHFSVRLLKFSREKKAAKTLGIVVGCFVLCWLPFFLVMPIGSFFPDFKPSETVFKIVFWLGYLNSCINPIIYPCSSQEFKKAFQNVLKIQCLRRKQSSKHALGYTLHPPSQAVEGQHKDMVRIPVGSRETFYKISKTDGVCEWKFFSSMPRGSARITVPKDQSACTTARVRSKSFLQVCCCVGPSTPNPGENHQVPTIKIHTISLSENGEEV