Target
Neuropeptide Y receptor type 1
Ligand
BDBM84999
Substrate
n/a
Ki
0.035±n/a nM
Comments
PDSP_3390
Citation
 Berglund, MMHolmberg, SKEriksson, HGedda, KMaffrand, JPSerradeil-Le Gal, CChhajlani, VGrundemar, LLarhammar, D The cloned guinea pig neuropeptide Y receptor Y1 conforms to other mammalian Y1 receptors. Peptides 20:1043-53 (1999) [PubMed]  Article 
Target
Name:
Neuropeptide Y receptor type 1
Synonyms:
NPY-Y1 | NPY1R | NPY1R_CAVPO
Type:
Enzyme Catalytic Domain
Mol. Mass.:
44288.14
Organism:
GUINEA PIG
Description:
NPY-Y1 NPY1R GUINEA PIG::Q9WVD0
Residue:
383
Sequence:
MNSTSFSQLENHSVHYNLSEEKPSFFAFENDDCHLPLAVIFTLALAYGAVIILGVSGNLALILIILKQKEMRNVTNILIVNLSFSDLLVAIMCLPFTFVYTLMDHWIFGEIMCKLNPFVQCVSITVSIFSLVLIAVERHQLIINPRGWRPNNRHAYIGIAVIWVLAVASSLPFMIYQVLTDEPFQNVTLDAFKDKLVCFDQFPSDSHRLSYTTLLLVLQYFGPLCFIFICYFKIYIRLKRRNNMMDKMRDSKYRSSESKRINIMLLSIVVAFAVCWLPLTIFNTVFDWNHQIIATCNHNLLFLLCHLTAMISTCVNPIFYGFLNKNFQRDLQFFFNFCDFRSRDDDYETIAMSTMHTDVSKTSLKQASPLAFKKISCVENEKI
  
Inhibitor
Name:
BDBM84999
Synonyms:
PYY,[leu31,Pro34], human
Type:
Small organic molecule
Emp. Form.:
C195H295N53O57
Mol. Mass.:
4293.7497
SMILES:
n/a
Structure:
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