Reaction Details Report a problem with these data
Target
Neurotensin receptor type 1
Ligand
BDBM82078
Substrate
n/a
Ki
0.25±n/a nM
Comments
PDSP_1308
Citation
Pettibone, DJ; Hess, JF; Hey, PJ; Jacobson, MA; Leviten, M; Lis, EV; Mallorga, PJ; Pascarella, DM; Snyder, MA; Williams, JB; Zeng, Z The effects of deleting the mouse neurotensin receptor NTR1 on central and peripheral responses to neurotensin. J Pharmacol Exp Ther 300:305-13 (2002) [PubMed] Article
More Info.:
Target
Name:
Neurotensin receptor type 1
Synonyms:
NT-R-1 | NTR1_MOUSE | Neurotensin 1 | Neurotensin receptor 1 | Neurotensin receptor type 1 | Ntsr | Ntsr1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
47237.04
Organism:
MOUSE
Description:
Neurotensin 1 NTSR1 MOUSE::A2ACT4
Residue:
424
Sequence:
MHLNSSVQQGAPSEPGAQPFPHPQFGLETMLLALSLSNGSGNSSESILEPNSNLDVNTDIYSKVLVTAVYLALFVVGTVGNSVTAFTLARKKSLQSLQSTVHYHLGSLALSDLLILLLAMPVELYNFIWVHHPWAFGDAGCRGYYFLRDACTYATALNVASLSVERYLAICHPFKAKTLMSRSRTKKFISAIWLASALLAVPMLFTMGLQNRSADGQHPGGLVCTPTVDTATVKVVIQVNTFMSFLFPMLIISILNTVIANKLTVMVHQAAEQGRGVCTVGTHNSLEHSTFNMSIEPGRVQALRHGVLVLRAVVIAFVVCWLPYHVRRLMFCYISDEQWTTFLFDFYHYFYMLTNALFYVSSAINPILYNLVSANFRQVFLSTLACLCPGWRRRRKKRPTFSRKPNSMSSNHAFSTSATRETLY