Reaction Details
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Report a problem with these dataTarget
Ionotropic glutamate receptor subunit Delta2
Ligand
BDBM86156
Substrate
n/a
Ki
>10000±n/a nM
Comments
PDSP_3022
Citation
Williams, K; Dattilo, M; Sabado, TN; Kashiwagi, K; Igarashi, K Pharmacology of delta2 glutamate receptors: effects of pentamidine and protons. J Pharmacol Exp Ther 305:740-8 (2003) [PubMed] Article More Info.:
Target
Name:
Ionotropic glutamate receptor subunit Delta2
Synonyms:
Glutamate delta 2 | Glutamate receptor delta-2 subunit
Type:
Enzyme Catalytic Domain
Mol. Mass.:
19076.25
Organism:
Xenopus
Description:
B9V8R6
Residue:
168
Sequence:
FDLSLWACIAGTVLLVGLLVYLLNWLNPPRLQMGSMTSTTLYNSMWFVYGSFVQQGGEVPYTTLATRMMMGAWWLFALIVISSYTANLAAFLTISRIESSIQSLQDLSRQTDIPYGTVFDSAVYEHVRVKGMNPFERDSMYSQMWRMINRSNGSENNVQESLEGIQKV
Inhibitor
Name:
BDBM86156
Synonyms:
CAS_3037648 | MB-3 | NSC_3037648
Type:
Small organic molecule
Emp. Form.:
C22H28N4O3S
Mol. Mass.:
428.548
SMILES:
CC(N(Cc1cnc(C)nc1N)C=O)=C(CCO)SCCC(=O)c1ccc(C)cc1 |w:1.0|
Structure:
