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Target
Melanocortin receptor 4
Ligand
BDBM88458
Substrate
n/a
Meas. Tech.
Luminescence-based cell-based high throughput dose response assay for biased ligands (agonists) of the melanocortin 4 receptor (MC4R)
EC50
>89215±n/a nM
Citation
 PubChem, PC Luminescence-based cell-based high throughput dose response assay for biased ligands (agonists) of the melanocortin 4 receptor (MC4R) PubChem Bioassay (2012)[AID] 
Target
Name:
Melanocortin receptor 4
Synonyms:
MC4-R | MC4R | MC4R_HUMAN | Melanocortin MC4 | Melanocortin receptor 4 (MC-4) | Melanocortin receptor 4 (MC4-R) | Melanocortin receptor 4 (MC4R)
Type:
Enzyme
Mol. Mass.:
36949.50
Organism:
Homo sapiens (Human)
Description:
P32245
Residue:
332
Sequence:
MVNSTHRGMHTSLHLWNRSSYRLHSNASESLGKGYSDGGCYEQLFVSPEVFVTLGVISLLENILVIVAIAKNKNLHSPMYFFICSLAVADMLVSVSNGSETIVITLLNSTDTDAQSFTVNIDNVIDSVICSSLLASICSLLSIAVDRYFTIFYALQYHNIMTVKRVGIIISCIWAACTVSGILFIIYSDSSAVIICLITMFFTMLALMASLYVHMFLMARLHIKRIAVLPGTGAIRQGANMKGAITLTILIGVFVVCWAPFFLHLIFYISCPQNPYCVCFMSHFNLYLILIMCNSIIDPLIYALRSQELRKTFKEIICCYPLGGLCDLSSRY
  
Inhibitor
Name:
BDBM88458
Synonyms:
2-[[[1-(4-chlorophenyl)-5-benzotriazolyl]amino]methylidene]propanedioic acid diethyl ester | 2-[[[1-(4-chlorophenyl)benzotriazol-5-yl]amino]methylene]malonic acid diethyl ester | MLS000698359 | SMR000224928 | cid_1827509 | diethyl 2-({[1-(4-chlorophenyl)-1H-1,2,3-benzotriazol-5-yl]amino}methylene)malonate | diethyl 2-[[[1-(4-chlorophenyl)benzotriazol-5-yl]amino]methylidene]propanedioate
Type:
Small organic molecule
Emp. Form.:
C20H19ClN4O4
Mol. Mass.:
414.842
SMILES:
[#6]-[#6]-[#8]-[#6](=O)-[#6](=[#6]\[#7]-c1ccc2n(nnc2c1)-c1ccc(Cl)cc1)\[#6](=O)-[#8]-[#6]-[#6]
Structure:
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