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Target
Melanocortin receptor 4
Ligand
BDBM88464
Substrate
n/a
Meas. Tech.
Luminescence-based cell-based high throughput dose response assay for biased ligands (agonists) of the melanocortin 4 receptor (MC4R)
EC50
>89181±n/a nM
Citation
 PubChem, PC Luminescence-based cell-based high throughput dose response assay for biased ligands (agonists) of the melanocortin 4 receptor (MC4R) PubChem Bioassay (2012)[AID] 
Target
Name:
Melanocortin receptor 4
Synonyms:
MC4-R | MC4R | MC4R_HUMAN | Melanocortin MC4 | Melanocortin receptor 4 (MC-4) | Melanocortin receptor 4 (MC4-R) | Melanocortin receptor 4 (MC4R)
Type:
Enzyme
Mol. Mass.:
36949.50
Organism:
Homo sapiens (Human)
Description:
P32245
Residue:
332
Sequence:
MVNSTHRGMHTSLHLWNRSSYRLHSNASESLGKGYSDGGCYEQLFVSPEVFVTLGVISLLENILVIVAIAKNKNLHSPMYFFICSLAVADMLVSVSNGSETIVITLLNSTDTDAQSFTVNIDNVIDSVICSSLLASICSLLSIAVDRYFTIFYALQYHNIMTVKRVGIIISCIWAACTVSGILFIIYSDSSAVIICLITMFFTMLALMASLYVHMFLMARLHIKRIAVLPGTGAIRQGANMKGAITLTILIGVFVVCWAPFFLHLIFYISCPQNPYCVCFMSHFNLYLILIMCNSIIDPLIYALRSQELRKTFKEIICCYPLGGLCDLSSRY
  
Inhibitor
Name:
BDBM88464
Synonyms:
(10Z)-10-[(4-hydroxyanilino)methylene]-8,8-dimethyl-pyrano[2,3-f]chromene-2,9-quinone | (10Z)-10-[(4-hydroxyanilino)methylidene]-8,8-dimethylpyrano[2,3-f][1]benzopyran-2,9-dione | (10Z)-10-[(4-hydroxyanilino)methylidene]-8,8-dimethylpyrano[2,3-f]chromene-2,9-dione | (10Z)-10-[[(4-hydroxyphenyl)amino]methylidene]-8,8-dimethyl-pyrano[2,3-f]chromene-2,9-dione | 10-{[(4-hydroxyphenyl)amino]methylene}-8,8-dimethyl-2H,8H-pyrano[2,3-f]chromene-2,9(10H)-dione | MLS000690659 | SMR000298918 | cid_2295134
Type:
Small organic molecule
Emp. Form.:
C21H17NO5
Mol. Mass.:
363.3634
SMILES:
CC1(C)Oc2ccc3ccc(=O)oc3c2C(=CNc2ccc(O)cc2)C1=O |w:16.18|
Structure:
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