Reaction Details Report a problem with these data
Target
Guanine nucleotide-binding protein subunit alpha-15
Ligand
BDBM96900
Substrate
n/a
EC50
>29910±n/a nM
Citation
 PubChem, PC Counterscreen for antagonists of the human trace amine associated receptor 1 (TAAR1): Fluorescence-based cell-based high throughput dose reponse assay to identify nonselective Ga16 agonists PubChem Bioassay (2013)[AID] 
Target
Name:
Guanine nucleotide-binding protein subunit alpha-15
Synonyms:
G protein alpha 16 | G-protein subunit alpha-16 | G-protein subunit alpha-16 (G alpha-16) | GNA15 | GNA15_HUMAN | GNA16 | Guanine nucleotide-binding protein subunit alpha-15 [Y147C]
Type:
Protein
Mol. Mass.:
43577.62
Organism:
Homo sapiens (Human)
Description:
P30679
Residue:
374
Sequence:
MARSLTWRCCPWCLTEDEKAAARVDQEINRILLEQKKQDRGELKLLLLGPGESGKSTFIKQMRIIHGAGYSEEERKGFRPLVYQNIFVSMRAMIEAMERLQIPFSRPESKHHASLVMSQDPYKVTTFEKRYAAAMQWLWRDAGIRACYERRREFHLLDSAVYYLSHLERITEEGYVPTAQDVLRSRMPTTGINEYCFSVQKTNLRIVDVGGQKSERKKWIHCFENVIALIYLASLSEYDQCLEENNQENRMKESLALFGTILELPWFKSTSVILFLNKTDILEEKIPTSHLATYFPSFQGPKQDAEAAKRFILDMYTRMYTGCVDGPEGSKKGARSRRLFSHYTCATDTQNIRKVFKDVRDSVLARYLDEINLL
  
Inhibitor
Name:
BDBM96900
Synonyms:
4-(1-oxopentylamino)-N-[4-(1-pyrrolidinylsulfonyl)phenyl]benzamide | 4-(pentanoylamino)-N-(4-pyrrolidin-1-ylsulfonylphenyl)benzamide | 4-(pentanoylamino)-N-[4-(1-pyrrolidinylsulfonyl)phenyl]benzamide | MLS000050100 | N-(4-pyrrolidinosulfonylphenyl)-4-(valerylamino)benzamide | SMR000077149 | cid_2957591
Type:
Small organic molecule
Emp. Form.:
C22H27N3O4S
Mol. Mass.:
429.532
SMILES:
CCCCC(=O)Nc1ccc(cc1)C(=O)Nc1ccc(cc1)S(=O)(=O)N1CCCC1
Structure:
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