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Target
Kallikrein-7
Ligand
BDBM90096
Substrate
n/a
EC50
6859±n/a nM
Citation
 PubChem, PC Fluorescence Intensity-based biochemical primary high throughput dose response assay to identify activators of kallikrein-7 (K7) zymogen PubChem Bioassay (2013)[AID] 
Target
Name:
Kallikrein-7
Synonyms:
KLK7 | KLK7_HUMAN | Kallikrein 7 | Kallikrein-7 | PRSS6 | SCCE | Serine protease 6 | Stratum corneum chymotryptic enzyme | hK7 | hSCCE | kallikrein-7 isoform 1 preproprotein
Type:
PROTEIN
Mol. Mass.:
27535.05
Organism:
Homo sapiens (Human)
Description:
ChEMBL_1469257
Residue:
253
Sequence:
MARSLLLPLQILLLSLALETAGEEAQGDKIIDGAPCARGSHPWQVALLSGNQLHCGGVLVNERWVLTAAHCKMNEYTVHLGSDTLGDRRAQRIKASKSFRHPGYSTQTHVNDLMLVKLNSQARLSSMVKKVRLPSRCEPPGTTCTVSGWGTTTSPDVTFPSDLMCVDVKLISPQDCTKVYKDLLENSMLCAGIPDSKKNACNGDSGGPLVCRGTLQGLVSWGTFPCGQPNDPGVYTQVCKFTKWINDTMKKHR
  
Inhibitor
Name:
BDBM90096
Synonyms:
MLS000578964 | SMR000198786 | butyl 3-(3-methylphenoxy)-4-oxo-4H-chromen-7-yl carbonate | butyl [3-(3-methylphenoxy)-4-oxidanylidene-chromen-7-yl] carbonate | butyl [3-(3-methylphenoxy)-4-oxochromen-7-yl] carbonate | carbonic acid butyl [3-(3-methylphenoxy)-4-oxo-1-benzopyran-7-yl] ester | carbonic acid butyl [4-keto-3-(3-methylphenoxy)chromen-7-yl] ester | cid_1638351
Type:
Small organic molecule
Emp. Form.:
C21H20O6
Mol. Mass.:
368.3799
SMILES:
CCCCOC(=O)Oc1ccc2c(c1)occ(Oc1cccc(C)c1)c2=O
Structure:
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