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Target
C-C motif chemokine 4
Ligand
BDBM633255
Substrate
n/a
Meas. Tech.
Biological and Stability Data
EC50
3.10±n/a nM
Citation
 Bazin-Lee, H; Ettenger, G; Khalaf, J; Ryter, KT Toll-like receptor ligands US Patent  US11458151 Publication Date 10/4/2022 
Target
Name:
C-C motif chemokine 4
Synonyms:
ACT-2 | CCL4 | CCL4_HUMAN | G-26 T-lymphocyte-secreted protein | HC21 | LAG-1 | LAG1 | Lymphocyte activation gene 1 protein | MIP-1-beta | MIP1B | Macrophage inflammatory protein 1-beta | PAT 744 | Protein H400 | SCYA4 | SIS-gamma | Small-inducible cytokine A4 | T-cell activation protein 2
Type:
Protein
Mol. Mass.:
10210.74
Organism:
Homo sapiens (Human)
Description:
P13236
Residue:
92
Sequence:
MKLCVTVLSLLMLVAAFCSPALSAPMGSDPPTACCFSYTARKLPRNFVVDYYETSSLCSQPAVVFQTKRSKQVCADPSESWVQEYVYDLELN
  
Inhibitor
Name:
BDBM633255
Synonyms:
GLA | Glycopyranoside Lipid A | MPLA | Monophosphoryl Lipid A | Monophosphoryl hexaacyl disaccharide | US11458151, Compound MPL
Type:
Small organic molecule
Emp. Form.:
C96H180N2O22P
Mol. Mass.:
1745.4309
SMILES:
CCCCCCCCCCCCCC(=O)O[C@H](CCCCCCCCCCC)CC(=O)N[C@H]1[C@H](OC[C@H]2O[C@H](O)[C@H](NC(=O)C[C@H](O)CCCCCCCCCCC)[C@@H](OC(=O)C[C@H](O)CCCCCCCCCCC)[C@@H]2O)O[C@H](CO)[C@@H](OP(O)([O-])=O)[C@@H]1OC(=O)C[C@@H](CCCCCCCCCCC)OC(=O)CCCCCCCCCCCCC
Structure:
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