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Target
Mitogen-activated protein kinase 1 [T157A]
Ligand
BDBM176675
Substrate
n/a
Meas. Tech.
Fluorescence Quenching Assay
Kd
3000±1000 nM
Citation
Shapiro, PS; MacKerell, Jr., AD; Fletcher, S Non-ATP dependent inhibitors of extracellular signal-regulated kinase (ERK) US Patent US9115122 Publication Date 8/25/2015
More Info.:
Target
Name:
Mitogen-activated protein kinase 1 [T157A]
Synonyms:
ERK2(T157A) | Erk2 | MK01_MOUSE | Mapk | Mapk1 | Prkm1
Type:
n/a
Mol. Mass.:
41248.63
Organism:
Mus musculus (Mouse)
Description:
P63085[T157A]
Residue:
358
Sequence:
MAAAAAAGPEMVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNLNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNATCDLKICDFGLARVADPDHDHTGFLTEYVATRWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFKFDMELDDLPKEKLKELIFEETARFQPGYRS