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Target
ELAV-like protein 1 [I180A]
Ligand
BDBM200223
Substrate
n/a
IC50
14700±n/a nM
Citation
 PubChem, PC Identify HuR specific inhibitors PubChem Bioassay (2015)[AID] 
Target
Name:
ELAV-like protein 1 [I180A]
Synonyms:
ELAV1_HUMAN | ELAVL1 | HUR | HuR RNA binding protein
Type:
Enzyme Catalytic Domain
Mol. Mass.:
36072.53
Organism:
Homo sapiens (Human)
Description:
gi_1022961
Residue:
326
Sequence:
MSNGYEDHMAEDCRGDIGRTNLIVNYLPQNMTQDELRSLFSSIGEVESAKLIRDKVAGHSLGYGFVNYVTAKDAERAINTLNGLRLQSKTIKVSYARPSSEVIKDANLYISGLPRTMTQKDVEDMFSRFGRIINSRVLVDQTTGLSRGVAFIRFDKRSEAEEAITSFNGHKPPGSSEPIAVKFAANPNQNKNVALLSQLYHSPARRFGGPVHHQAQRFRFSPMGVDHMSGLSGVNVPGNASSGWCIFIYNLGQDADEGILWQMFGPFGAVTNVKVIRDFNTNKCKGFGFVTMTNYEEAAMAIASLNGYRLGDKILQVSFKTNKSHK
  
Inhibitor
Name:
BDBM200223
Synonyms:
cid_3034178
Type:
Small organic molecule
Emp. Form.:
C17H18N2O3S2
Mol. Mass.:
362.466
SMILES:
CC1=CC(C)(C)NC(=S)N1c1cccc2cc(ccc12)S(O)(=O)=O |t:1|
Structure:
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