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Target
ELAV-like protein 1 [I180A]
Ligand
BDBM200225
Substrate
n/a
IC50
2700±n/a nM
Citation
 PubChem, PC Identify HuR specific inhibitors PubChem Bioassay (2015)[AID] 
Target
Name:
ELAV-like protein 1 [I180A]
Synonyms:
ELAV1_HUMAN | ELAVL1 | HUR | HuR RNA binding protein
Type:
Enzyme Catalytic Domain
Mol. Mass.:
36072.53
Organism:
Homo sapiens (Human)
Description:
gi_1022961
Residue:
326
Sequence:
MSNGYEDHMAEDCRGDIGRTNLIVNYLPQNMTQDELRSLFSSIGEVESAKLIRDKVAGHSLGYGFVNYVTAKDAERAINTLNGLRLQSKTIKVSYARPSSEVIKDANLYISGLPRTMTQKDVEDMFSRFGRIINSRVLVDQTTGLSRGVAFIRFDKRSEAEEAITSFNGHKPPGSSEPIAVKFAANPNQNKNVALLSQLYHSPARRFGGPVHHQAQRFRFSPMGVDHMSGLSGVNVPGNASSGWCIFIYNLGQDADEGILWQMFGPFGAVTNVKVIRDFNTNKCKGFGFVTMTNYEEAAMAIASLNGYRLGDKILQVSFKTNKSHK
  
Inhibitor
Name:
BDBM200225
Synonyms:
cid_5992379
Type:
Small organic molecule
Emp. Form.:
C11H12AsN5O4S
Mol. Mass.:
385.231
SMILES:
CSC1=NC(=O)\C(=N/Nc2ccc(cc2)[As](O)(O)=O)C(N)=N1 |c:21,t:2|
Structure:
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