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Target
TspO-like protein
Ligand
BDBM209869
Substrate
n/a
Meas. Tech.
Tryptophan Fluorescence Assay
Kd
4.63e+3±n/a nM
Citation
 Busch, AW; WareJoncas, Z; Montgomery, BL Tryptophan-Rich Sensory Protein/Translocator Protein (TSPO) from Cyanobacterium Fremyella diplosiphon Binds a Broad Range of Functionally Relevant Tetrapyrroles. Biochemistry 56:73-84 (2017) [PubMed]  Article 
Target
Name:
TspO-like protein
Synonyms:
Tryptophan-rich sensory protein/translocator protein (TSPO)
Type:
Protein
Mol. Mass.:
28330.64
Organism:
Fremyella diplosiphon (Cyanobacterium)
Description:
Q6GZK8
Residue:
251
Sequence:
MTQSNNTGILEKFVNTVMGVKTENQQQPSNTLIATTQALDIRAVLVYKLGTILQIAAMMLALLGMEKLVMLIDKNSHLPSWFSTLLAVLFFALLSIRSRIFSLLDNTRSRKTYDQVIRPRWAPPPLVFPIVWMIIAVLRVISSVLIWQQMHHQFLALPLILFVVHLALGDTWNTIFTVERRLGAAVPVVILGPWLSALVVTAIYWQTNPVAGMIFSFSCIWLTVAAVLVFRIWQLNGSEPLYPLKLTPVEK
  
Inhibitor
Name:
BDBM209869
Synonyms:
3-[(2E,5E)-2-[[3-(2-carboxyethyl)-5-[(E)-(3-ethenyl-4-methyl-5-oxopyrrol-2-ylidene)methyl]-4-methyl-1H-pyrrol-2-yl]methylidene]-5-[(4-ethenyl-3-methyl-5-oxopyrrol-2-yl)methylidene]-4-methylpyrrol-3-yl]propanoic acid | Biliverdin IXα
Type:
Small organic molecule
Emp. Form.:
C33H34N4O6
Mol. Mass.:
582.6463
SMILES:
CC1=C(C=C)\C(NC1=O)=C/c1[nH]c(\C=c2\[nH]\c(=C\C3=NC(=O)C(C=C)=C3C)c(C)c2CCC(O)=O)c(CCC(O)=O)c1C |c:1,25,t:19|
Structure:
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