Reaction Details Report a problem with these data
Target
Growth hormone secretagogue receptor type 1 [E24Q]
Ligand
BDBM212437
Substrate
n/a
Meas. Tech.
GHS Ligand Binding Assay
Ki
915±0 nM
Citation
Mary, S; Fehrentz, JA; Damian, M; Gaibelet, G; Orcel, H; Verdié, P; Mouillac, B; Martinez, J; Marie, J; Banères, JL Heterodimerization with Its splice variant blocks the ghrelin receptor 1a in a non-signaling conformation: a study with a purified heterodimer assembled into lipid discs. J Biol Chem 288:24656-65 (2013) [PubMed] Article
More Info.:
Target
Name:
Growth hormone secretagogue receptor type 1 [E24Q]
Synonyms:
GHSR | GHSR_HUMAN | Ghrelin receptor 1a (GHS-R1a E124Q)
Type:
Protein
Mol. Mass.:
41334.59
Organism:
Homo sapiens (Human)
Description:
Human ghrelin receptor 1a E124Q mutant
Residue:
366
Sequence:
MWNATPSEEPGFNLTLADLDWDASPGNDSLGDELLQLFPAPLLAGVTATCVALFVVGIAGNLLTMLVVSRFRELRTTTNLYLSSMAFSDLLIFLCMPLDLVRLWQYRPWNFGDLLCKLFQFVSQSCTYATVLTITALSVERYFAICFPLRAKVVVTKGRVKLVIFVIWAVAFCSAGPIFVLVGVEHENGTDPWDTNECRPTEFAVRSGLLTVMVWVSSIFFFLPVFCLTVLYSLIGRKLWRRRRGDAVVGASLRDQNHKQTVKMLAVVVFAFILCWLPFHVGRYLFSKSFEPGSLEIAQISQYCNLVSFVLFYLSAAINPILYNIMSKKYRVAVFRLLGFEPFSQRKLSTLKDESSRAWTESSINT