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Target
BioDB n*138 SEQ ID NO: 2
Ligand
BDBM239075
Substrate
n/a
Meas. Tech.
Functional Assay
IC50
225±n/a nM
Citation
 Prather, PL; Prisinzano, TE; Fantegrossi, WE; Brents, LK; Moran, J; Radominska-Pandya, A; Vasiljevik, T Use of the aminoalkylindole JWH-073-M4 and related compounds as neutral CB1 receptor antagonists for the treatment of alcoholism, drug abuse, obesity, and obesity-related diseases US Patent  US9416103 Publication Date 8/16/2016 
Target
Name:
BioDB n*138 SEQ ID NO: 2
Synonyms:
n/a
Type:
Peptide Substrate
Mol. Mass.:
3822.64
Organism:
Artificial Organism
Description:
SEQ ID NO: 2
Residue:
30
Sequence:
KWEEINGNNYVYIDPTQLPYDHKWEFPRNR
  
Inhibitor
Name:
BDBM239075
Synonyms:
US9416103, JWH-073-M4
Type:
Small organic molecule
Emp. Form.:
C23H21NO2
Mol. Mass.:
343.4183
SMILES:
CCCCn1cc(C(=O)c2cccc3ccccc23)c2cccc(O)c12
Structure:
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