Reaction Details Report a problem with these data
Target
Cannabinoid receptor 2
Ligand
BDBM239141
Substrate
n/a
Meas. Tech.
Cannabinoid Receptor Binding Assay
Ki
>1.0e+4±n/a nM
IC50
>1.0e+4±n/a nM
Citation
 Taher, AT; Kadry, HH; Allarà, M; Di Marzo, V; Abadi, AH; Abouzid, KA Synthesis and binding study of certain 6-arylalkanamides as molecular probes for cannabinoid receptor subtypes. J Enzyme Inhib Med Chem 28:436-9 (2013) [PubMed]  Article 
Target
Name:
Cannabinoid receptor 2
Synonyms:
CANNABINOID CB2 | CB-2 | CB2 | CB2A | CB2B | CNR2 | CNR2_HUMAN | CX5 | Cannabinoid CB2 receptor | Cannabinoid receptor 2 (CB2) | Cannabinoid receptor 2 (CB2R) | hCB2
Type:
G Protein-Coupled Receptor (GPCR)
Mol. Mass.:
39690.94
Organism:
Homo sapiens (Human)
Description:
P34972
Residue:
360
Sequence:
MEECWVTEIANGSKDGLDSNPMKDYMILSGPQKTAVAVLCTLLGLLSALENVAVLYLILSSHQLRRKPSYLFIGSLAGADFLASVVFACSFVNFHVFHGVDSKAVFLLKIGSVTMTFTASVGSLLLTAIDRYLCLRYPPSYKALLTRGRALVTLGIMWVLSALVSYLPLMGWTCCPRPCSELFPLIPNDYLLSWLLFIAFLFSGIIYTYGHVLWKAHQHVASLSGHQDRQVPGMARMRLDVRLAKTLGLVLAVLLICWFPVLALMAHSLATTLSDQVKKAFAFCSMLCLINSMVNPVIYALRSGEIRSSAHHCLAHWKKCVRGLGSEAKEEAPRSSVTETEADGKITPWPDSRDLDLSDC
  
Inhibitor
Name:
BDBM239141
Synonyms:
(E) Ethyl [2-(4-oxo-6-phenylhex)-5-enamido]acetate (3c)
Type:
Small organic molecule
Emp. Form.:
C13H15NO3
Mol. Mass.:
233.2631
SMILES:
CCOC(=O)CNC(=O)\C=C\c1ccccc1
Structure:
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