Reaction Details Report a problem with these data
Target
Somatostatin receptor type 2
Ligand
BDBM275984
Substrate
n/a
Meas. Tech.
Radioligand Binding Assays
Ki
9630±n/a nM
Citation
 Mazzaferro, R; Ferrara, M; Giovannini, R; Lingard, I; Rudolf, K Morpholine and 1,4-oxazepane amides as somatostatin receptor subtype 4 (SSTR4) agonists US Patent  US10577336 Publication Date 3/3/2020 
Target
Name:
Somatostatin receptor type 2
Synonyms:
SOMATOSTATIN SST2 | SRIF-1 | SS-2-R | SS2-R | SS2R | SSR2_HUMAN | SSTR2 | Somatostatin receptor type 2 (SSTR2)
Type:
Enzyme
Mol. Mass.:
41344.94
Organism:
Homo sapiens (Human)
Description:
P30874
Residue:
369
Sequence:
MDMADEPLNGSHTWLSIPFDLNGSVVSTNTSNQTEPYYDLTSNAVLTFIYFVVCIIGLCGNTLVIYVILRYAKMKTITNIYILNLAIADELFMLGLPFLAMQVALVHWPFGKAICRVVMTVDGINQFTSIFCLTVMSIDRYLAVVHPIKSAKWRRPRTAKMITMAVWGVSLLVILPIMIYAGLRSNQWGRSSCTINWPGESGAWYTGFIIYTFILGFLVPLTIICLCYLFIIIKVKSSGIRVGSSKRKKSEKKVTRMVSIVVAVFIFCWLPFYIFNVSSVSMAISPTPALKGMFDFVVVLTYANSCANPILYAFLSDNFKKSFQNVLCLVKVSGTDDGERSDSKQDKSRLNETTETQRTLLNGDLQTSI
  
Inhibitor
Name:
BDBM275984
Synonyms:
US10071974, Example 95 | US10577336, Example 95
Type:
Small organic molecule
Emp. Form.:
C16H22N4O2
Mol. Mass.:
302.3715
SMILES:
Cc1cccn2c(ncc12)C(C)(C)NC(=O)[C@@H]1CNCCO1 |r|
Structure:
Search PDB for entries with ligand similarity: