Assay Method Information | |
| ChEMBL_978570 (CHEMBL2421940) |
Description: | Antagonist activity at CB2 receptor in HEK293 cells assessed as increase in CP-55,940 EC50 measuring inhibition of forskolin-stimulated cAMP accumulation at 1 uM incubated 20 mins prior to CP-55,940 addition measured after 7 mins by spectrophotometry (Rvb = 4.21+/-1.16 nM) |
Affinity data for this assay | |
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