Assay Method Information

Assay Name:  ChEMBL_1908813 (CHEMBL4411171)
Description:  Inhibition of 0.05 nM DOT1L (2 to 416 residues) (unknown origin) using biotinylated nucleosome as substrate and [3H]SAM as co-factor preincubated for 30 mins followed by substrate and cofactor addition and measured after 180 mins by scintillation proximity assay
Affinity data for this assay
 

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