Assay Method Information

Assay Name:  ChEMBL_2185269 (CHEMBL5097351)
Description:  Inhibition of recombinant N-terminal MBP-tagged human PLK3-PBD expressed in Escherichia coli BL21(DE3) rosetta cells using 5-carboxyfluorescein-GPLATSpTPKNG-NH2 as substrate preincubated for 1 hr followed by substrate addition and measured after 1 hr by fluorescence polarization assay
Affinity data for this assay
 

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