Assay Method Information

Assay Name:  ChEMBL_2213078 (CHEMBL5126027)
Description:  Antagonist activity at human MRGPRX2 expressed in HEK293 cells co-expressing mouse Galpha15 assessed as inhibition of Cortistatin-14 induced Ca2+ mobilization preincubated for 30 mins followed by Cortistatin-14 addition by FLIPRtetra-calcium mobilization assay
Affinity data for this assay
 

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