Assay Method Information

Assay Name:  ChEMBL_2435320
Description:  Displacement of kinase tracer 236 from ATP-binding site of biotinylated N-terminal TEV-fused/hexahistidine tagged C-terminal avidin tagged human DYRK1A kinase domain (127 to 485 residues) transfected in Escherichia coli BL21 (DE3)-R3 incubated for 1.5 hrs by TR-FRET assay
Affinity data for this assay
 

If you find an error in this entry please send us an E-mail