| Assay Method Information | |
| | ChEMBL_2453378 |
| Description: | Antagonist activity at AR in human LNCaP cells assessed as reduction in R1881-induced AR transcriptional activity preincubated for 60 mins followed by R1881 addition and measured after 24 hrs by Steady-Glo reagent based luciferase assay |
| Affinity data for this assay | |
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