| Assay Method Information | |
| | ChEMBL_2453670 |
| Description: | Noncompetitive inhibition of epibatidine-induced receptor activation at rat alpha3beta4 nAChR expressed in HEK293 cells assessed as reduction in calcium flux by measuring increase in EC50 pretreated with compound for 10 mins followed by epibatidine addition and measured for 90 secs by FLIPR assay (Rvb = 320 nM) |
| Affinity data for this assay | |
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