Assay Method Information

Assay Name:  ChEMBL_1661643 (CHEMBL4011255)
Description:  Antagonist activity at human P2Y12 receptor expressed in CHO cells assessed as inhibition of 2-MeSADP-induced beta-arrestin translocation preincubated for 30 mins followed by 2-MeSADP addition measured after 90 mins by luminescence-based topcount method
Affinity data for this assay
 

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