Assay Method Information

Assay Name:  ChEMBL_2046327 (CHEMBL4701026)
Description:  Antagonist activity at human adenosine 2A receptor expressed in HEK293 cells assessed as reduction in cAMP production preincubated for 10 mins followed by 3 nM A2A agonist NECA addition and measured after 30 mins by EU-cAMP tracer based TR-FRET assay
Affinity data for this assay
 

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