| Assay Method Information | |
| | ChEMBL_2123255 (CHEMBL4832488) |
| Description: | Positive allosteric modulator activity in mouse kappa opioid receptor stably expressed in HEK293 cell membrane assessed as inhibition of forskolin induced cAMP production by measuring U50,488 EC50 at 3 uM pretreated for 30 mins followed by coincubation with U50,488 measured after 30 mins by HTRF assay |
| Affinity data for this assay | |
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