| Assay Method Information | |
| | ChEMBL_2496609 |
| Description: | Antagonist activity at human CAR LBD (151 to 349 residues) expressed in HepG2 cells co-expressed with pGL5-luc luciferase assessed as reduction in CAR activation measured after 1 to 4 hrs by LanthaScreen TR-FRET assay |
| Affinity data for this assay | |
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