Assay Method Information

Assay Name:  ChEMBL_2185274 (CHEMBL5097356)
Description:  Inhibition of human PLK1-PBD expressed in Escherichia coli BL21(DE3) rosetta cells using 5-carboxyfluorescein-GPMQSpTPLNG-OH as substrate preincubated for 1 hr followed by substrate addition and measured after 1 hr by fluorescence polarization assay
Affinity data for this assay
 

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