Assay Method Information

Assay Name:  ChEMBL_2207453 (CHEMBL5120161)
Description:  Antagonist activity at human P2X7 receptor expressed in HEK293 cells assessed as reduction in YO-PRO-1 iodide dye uptake preincubated for 30 mins followed by YO-PRO-1 iodide addition and measured after 120 mins by fluorescence plate reader analysis
Affinity data for this assay
 

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