| Assay Method Information | |
| | ChEMBL_2185275 (CHEMBL5097357) |
| Description: | Inhibition of recombinant C-terminal 6His-tagged human PLK2-PBD expressed in Escherichia coli BL21(DE3) rosetta cells using 5-carboxyfluorescein-GPMQTSpTPKNG-OH as substrate preincubated for 1 hr followed by substrate addition and measured after 1 hr by fluorescence polarization assay |
| Affinity data for this assay | |
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