Assay Method Information

Assay Name:  ChEMBL_1634655 (CHEMBL3877553)
Description:  Antagonist activity at human alpha4beta2 expressed in human SH-EP1 cells assessed as reduction in carbamylcholine induced 86Rb+ efflux preincubated for 10 mins followed by carbamylcholine addition measured after 5 mins by Cherenkov counting
Affinity data for this assay
 

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