Compile Data Set for Download or QSAR
Report error Found 31 of affinity data for UniProtKB/TrEMBL: A0A0D9RHK8
TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354702BDBM354702(US9809583, Example 10 | t-butyl(4-hydroxybenzyl)ca...)
Affinity DataIC50: 6.30nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354706BDBM354706(US9809583, Example 19 | 4-((2R,5S)-5-((4-cyanophen...)
Affinity DataIC50: 7.60nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354712BDBM354712(US9809583, Example 25 | N-(4-(((2R,5S)-3-(4-cyano-...)
Affinity DataIC50: 8.5nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354721BDBM354721(US9809583, Example 33 | ((2S,5S)-3-(3-methyl-4-nit...)
Affinity DataIC50: 10.4nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354703BDBM354703(US9809583, Example 11 | 4-((2R,5S)-5-((4-cyano-2-f...)
Affinity DataIC50: 10.5nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354698BDBM354698(US9809583, Example 6 | ((2R,5S)-3-(3-methyl-4-nitr...)
Affinity DataIC50: 11nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354700BDBM354700(US9809583, Example 8 | ((2R,5S)-3-(3-trifluorometh...)
Affinity DataIC50: 13.7nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354719BDBM354719(US9809583, Example 31 | 4-(2R,5S)-5-((3-fluoro-4-n...)
Affinity DataIC50: 14.1nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354717BDBM354717(US9809583, Example 29 | (S)-2-hydroxy-3-((4-nitro-...)
Affinity DataIC50: 14.1nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354705BDBM354705(US9809583, Example 13 | (S)-3-((4-cyano-3-(trifluo...)
Affinity DataIC50: 14.5nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354699BDBM354699(US9809583, Example 7 | (S)-3-((4-nitro-3-(trifluor...)
Affinity DataIC50: 15.7nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354715BDBM354715(US9809583, Example 27 | 4-((2R,5S)-5-((4-methoxyph...)
Affinity DataIC50: 22.4nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354694BDBM354694(US9809583, Example 2 | 4-((2S,5S)-5-(hydroxymethyl...)
Affinity DataIC50: 23.9nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354722BDBM354722(US9809583, Example 34 | 4-(((2R,5S)-3-(4-cyano-3-(...)
Affinity DataIC50: 24.1nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354720BDBM354720(US9809583, Example 32 | (2R,5S)-3-(4-nitro-3-(trif...)
Affinity DataIC50: 32.7nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354714BDBM354714(US9809583, Example 26 | ethyl(S)-3-((3-chloro-4-ni...)
Affinity DataIC50: 43.6nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354710BDBM354710(US9809583, Example 23 | 4-((2R,5S)-5-((R)-2,2,2-tr...)
Affinity DataIC50: 44.3nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354693BDBM354693(US9809583, Example 1 | (S)-4-((2,3-dihydroxypropyl...)
Affinity DataIC50: 64.4nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354713BDBM354713(US9809583, Example 56 | 4-((2R,5S)-5-((4-chlorophe...)
Affinity DataIC50: 75.1nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354716BDBM354716(US9809583, Example 28 | 4-((2R,5S)-5-((3-methoxyph...)
Affinity DataIC50: 77.2nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354697BDBM354697(US9809583, Example 5 | 4-((2R,5R)-5-((4-cyanopheno...)
Affinity DataIC50: 91.6nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354711BDBM354711(US9809583, Example 24 | (2R,5S)-3-(3-methyl-4-nitr...)
Affinity DataIC50: 141nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354718BDBM354718(US9809583, Example 30 | N-(4-(((2S,5S)-3-(4-cyano-...)
Affinity DataIC50: 142nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354704BDBM354704(US9809583, Example 12 | 4-((2R,5R)-5-(aminomethyl)...)
Affinity DataIC50: 145nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354723BDBM354723(US9809583, Example 35 | 4-((2S,5S)-5-((4-nitrophen...)
Affinity DataIC50: 185nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354701BDBM354701(US9809583, Example 9 | 4-(((2R,5S)-3-(4-cyano-3-(t...)
Affinity DataIC50: 367nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354696BDBM354696(US9809583, Example 4 | (S)-3-((3-methyl-4-nitrophe...)
Affinity DataIC50: 657nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354708BDBM354708(US9809583, Example 21 | 4-((2S,5R)-5-((R)-2,2,2-tr...)
Affinity DataIC50: 1.06E+3nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354707BDBM354707(US9809583, Example 20 | 4-((2S,5R)-5-((4-cyanophen...)
Affinity DataIC50: 1.08E+3nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354695BDBM354695(US9809583, Example 3 | 4-((2S,5R)-5-(hydroxymethyl...)
Affinity DataIC50: 1.09E+3nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354709BDBM354709(US9809583, Example 22 | 4-((2S,5R)-5-((S)-2,2,2-tr...)
Affinity DataIC50: 1.87E+3nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent