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TargetPhosphoglycerate kinase 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50643622(CHEMBL4528432)
Affinity DataKd:  2.10nMAssay Description:Binding affinity to PGK1 (unknown origin) exogenously expressed in Escherichia coli assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50587785(CHEMBL5178368)
Affinity DataKd:  3.70nMAssay Description:Binding affinity to PGK1 (unknown origin) exogenously expressed in Escherichia coli assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50652793(CHEMBL5653589)
Affinity DataKd:  57nMAssay Description:Binding affinity to human PGK1 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50216719(CHEMBL348433)
Affinity DataKi:  330nMpH: 7.1Assay Description:Binding affinity was evaluated towards 3-phosphoglycerate kinase at 37 degrees Celsius in 0.1 m NaCl pH 7.1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50216635(CHEMBL356436)
Affinity DataKi:  690nMpH: 7.1Assay Description:Binding affinity was evaluated towards 3-phosphoglycerate kinase at 37 degrees Celsius in 0.1 m NaCl pH 7.1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50216704(CHEMBL150751)
Affinity DataIC50: 840nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50216708(CHEMBL151887)
Affinity DataIC50: 880nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50216723(CHEMBL150369)
Affinity DataIC50: 960nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50216696(CHEMBL357952)
Affinity DataIC50: 980nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50216716(CHEMBL348186)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50216634(CHEMBL356655)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50216714(CHEMBL149734)
Affinity DataIC50: 1.08E+3nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50216726(CHEMBL149786)
Affinity DataIC50: 1.15E+3nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50216701(CHEMBL148974)
Affinity DataIC50: 1.17E+3nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50216635(CHEMBL356436)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50216719(CHEMBL348433)
Affinity DataIC50: 1.34E+3nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50216707(CHEMBL422133)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50216636(CHEMBL347337)
Affinity DataIC50: 1.98E+3nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50469690(CHEMBL85343)
Affinity DataKd:  2.00E+3nMAssay Description:Equilibrium binding affinity against histamine-62 residue of phosphoglycerokinase in yeastMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2020
Entry Details Article

TargetPhosphoglycerate kinase 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50216700(CHEMBL149264)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50469690(CHEMBL85343)
Affinity DataKd:  4.00E+3nMAssay Description:Equilibrium binding affinity against histamine-167 residue of phosphoglycerokinase in yeastMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2020
Entry Details Article

TargetPhosphoglycerate kinase 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50469693(CHEMBL88020)
Affinity DataKd:  4.00E+3nMAssay Description:Equilibrium binding affinity against histamine-167 residue of phosphoglycerokinase in yeastMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2020
Entry Details Article

TargetPhosphoglycerate kinase 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50652792(CHEMBL3752910)
Affinity DataKd:  5.21E+3nMAssay Description:Binding affinity to human PGK1 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetPhosphoglycerate kinase 1/2(Human)
University of Sheffield

Curated by ChEMBL
LigandPNGBDBM50216217(CHEMBL1160562)
Affinity DataKd:  6.00E+3nMAssay Description:Dissociation constant for binding with Phosphoglycerate kinase (PGK) enzyme is evaluatedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50469693(CHEMBL88020)
Affinity DataKd:  7.00E+3nMAssay Description:Equilibrium binding affinity against histamine-170 residue of phosphoglycerokinase in yeastMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2020
Entry Details Article

TargetPhosphoglycerate kinase 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50469690(CHEMBL85343)
Affinity DataKd:  7.00E+3nMAssay Description:Equilibrium binding affinity against histamine-170 residue of phosphoglycerokinase in yeastMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2020
Entry Details Article

TargetPhosphoglycerate kinase 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50216722(CHEMBL149115)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50469693(CHEMBL88020)
Affinity DataKd:  8.00E+3nMAssay Description:Equilibrium binding affinity against histamine-62 residue of phosphoglycerokinase in yeastMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2020
Entry Details Article

TargetPhosphoglycerate kinase 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50216695(CHEMBL149058)
Affinity DataIC50: 8.35E+3nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50216679(CHEMBL149129)
Affinity DataIC50: 9.40E+3nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50216710(CHEMBL345538)
Affinity DataIC50: 1.07E+4nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50216222(CHEMBL609443)
Affinity DataKd:  1.30E+4nMAssay Description:Dissociation constant for binding with Phosphoglycerate kinase (PGK) enzyme is evaluatedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50216720(CHEMBL149998)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50216705(CHEMBL149943)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50367883(CHEMBL605451)
Affinity DataIC50: 3.00E+4nMAssay Description:evaluated for the inhibition of Trypanosoma brucei Phosphoglycerate kinase (PGK)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50472926(CHEMBL607503)
Affinity DataIC50: 5.00E+4nMAssay Description:evaluated for the inhibition of Trypanosoma brucei Phosphoglycerate kinase (PGK)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50216724(CHEMBL356430)
Affinity DataKi:  6.10E+4nMpH: 7.1Assay Description:Binding affinity was evaluated towards 3-phosphoglycerate kinase at 37 degrees Celsius in 0.1 m NaCl pH 7.1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50216699(CHEMBL147415)
Affinity DataKi:  6.10E+4nMpH: 7.1Assay Description:Binding affinity was evaluated towards 3-phosphoglycerate kinase at 37 degrees Celsius in 0.1 m NaCl pH 7.1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50469692(CHEMBL87319)
Affinity DataKd:  6.60E+4nMAssay Description:Equilibrium binding affinity against histamine-170 residue of phosphoglycerokinase in yeastMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2020
Entry Details Article

TargetPhosphoglycerate kinase 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50216709(CHEMBL148780)
Affinity DataIC50: 6.88E+4nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50469692(CHEMBL87319)
Affinity DataKd:  7.10E+4nMAssay Description:Equilibrium binding affinity against histamine-167 residue of phosphoglycerokinase in yeastMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2020
Entry Details Article

TargetPhosphoglycerate kinase 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50216702(CHEMBL148792)
Affinity DataIC50: 7.30E+4nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50216698(CHEMBL341829)
Affinity DataKi:  7.50E+4nMpH: 7.1Assay Description:Binding affinity was evaluated towards 3-phosphoglycerate kinase at 37 degrees Celsius in 0.1 m NaCl pH 7.1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50216717(CHEMBL149729)
Affinity DataIC50: 7.80E+4nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50469692(CHEMBL87319)
Affinity DataKd:  8.00E+4nMAssay Description:Equilibrium binding affinity against histamine-62 residue of phosphoglycerokinase in yeastMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2020
Entry Details Article

TargetPhosphoglycerate kinase 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50216703(CHEMBL148705)
Affinity DataKi:  8.00E+4nMpH: 7.1Assay Description:Binding affinity was evaluated towards 3-phosphoglycerate kinase at 37 degrees Celsius in 0.1 m NaCl pH 7.1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50216724(CHEMBL356430)
Affinity DataIC50: 8.70E+4nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50216699(CHEMBL147415)
Affinity DataIC50: 8.70E+4nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50216713(CHEMBL345282)
Affinity DataIC50: 8.90E+4nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50469695(CHEMBL87788 | CHEBI:17050)
Affinity DataKd:  9.40E+4nMAssay Description:Equilibrium binding affinity against histamine-167 residue of phosphoglycerokinase in yeastMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2020
Entry Details Article
PDB3D3D Structure (crystal)
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