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Report error Found 174 of affinity data for UniProtKB/TrEMBL: P00730
TargetCarboxypeptidase A1(Bovine)
University of Athens

LigandPNGBDBM21471(2-benzyl-3-{[1-(2-acetamido-4-methylpentanamido)-2...)
Affinity DataKi:  0.300nMAssay Description:Continuous assays were performed by recording the fluorescence increase at 405 nm (excitation@ 320 nm) induced by the cleavage of fluorogenic substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2008
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
University of Athens

LigandPNGBDBM21464(The second fraction of the HPLC chromatogram. | 2-...)
Affinity DataKi:  0.5nMAssay Description:Continuous assays were performed by recording the fluorescence increase at 405 nm (excitation@ 320 nm) induced by the cleavage of fluorogenic substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2008
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
University of Athens

LigandPNGBDBM50109593(SQ-14603 | 2-Mercaptomethyl-3-phenyl-propionic aci...)
Affinity DataKi:  10nMAssay Description:Inhibition of bovine carboxypeptidase A (CPA) using hippuryl-L-phenylalanine (Hipp-L-Phe) as a substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
University of Athens

LigandPNGBDBM50109593(SQ-14603 | 2-Mercaptomethyl-3-phenyl-propionic aci...)
Affinity DataKi:  11nMAssay Description:Compound was evaluated for binding affinity against carboxypeptidase A (CPA), expressed as inhibitory constant (Ki)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCarboxypeptidase A1(Bovine)
University of Athens

LigandPNGBDBM50109593(SQ-14603 | 2-Mercaptomethyl-3-phenyl-propionic aci...)
Affinity DataKi:  11nMAssay Description:Binding affinity against carboxypeptidase A using hippurylphenylalanine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCarboxypeptidase A1(Bovine)
University of Athens

LigandPNGBDBM50109593(SQ-14603 | 2-Mercaptomethyl-3-phenyl-propionic aci...)
Affinity DataKi:  11nMAssay Description:Inhibition of bovine pancreatic carboxypeptidase AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
University of Athens

LigandPNGBDBM50279954(3-(3-Fluoro-phenyl)-2-mercaptomethyl-propionic aci...)
Affinity DataKi:  35nMAssay Description:Binding affinity against carboxypeptidase A using hippurylphenylalanine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCarboxypeptidase A1(Bovine)
University of Athens

LigandPNGBDBM21473(3-{[1-(2-acetamido-4-methylpentanoyl)pyrrolidin-2-...)
Affinity DataKi:  35nMAssay Description:Continuous assays were performed by recording the fluorescence increase at 405 nm (excitation@ 320 nm) induced by the cleavage of fluorogenic substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2008
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
University of Athens

LigandPNGBDBM50279947(3-(4-Fluoro-phenyl)-2-mercaptomethyl-propionic aci...)
Affinity DataKi:  37nMAssay Description:Compound was evaluated for binding affinity against carboxypeptidase A (CPA), expressed as inhibitory constant (Ki)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCarboxypeptidase A1(Bovine)
University of Athens

LigandPNGBDBM50279947(3-(4-Fluoro-phenyl)-2-mercaptomethyl-propionic aci...)
Affinity DataKi:  37nMAssay Description:Binding affinity against carboxypeptidase A using hippurylphenylalanine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCarboxypeptidase A1(Bovine)
University of Athens

LigandPNGBDBM50279958(3-(2-Fluoro-phenyl)-2-mercaptomethyl-propionic aci...)
Affinity DataKi:  45nMAssay Description:Binding affinity against carboxypeptidase A using hippurylphenylalanine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCarboxypeptidase A1(Bovine)
University of Athens

LigandPNGBDBM50109588((S)3-Mercapto-2-phenethylamino-propionic acid | CH...)
Affinity DataKi:  55nMAssay Description:Inhibition of bovine carboxypeptidase A (CPA) using hippuryl-L-phenylalanine (Hipp-L-Phe) as a substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
University of Athens

LigandPNGBDBM21470(The second fraction of the HPLC chromatogram. | 2-...)
Affinity DataKi:  60nMAssay Description:Continuous assays were performed by recording the fluorescence increase at 405 nm (excitation@ 320 nm) induced by the cleavage of fluorogenic substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2008
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
University of Athens

LigandPNGBDBM50109585(3-Mercapto-2-phenethylamino-propionic acid | CHEMB...)
Affinity DataKi:  65nMAssay Description:Inhibition of bovine carboxypeptidase A (CPA) using hippuryl-L-phenylalanine (Hipp-L-Phe) as a substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
University of Athens

LigandPNGBDBM50279960(2-Mercaptomethyl-3-phenyl-butyric acid | CHEMBL109...)
Affinity DataKi:  105nMAssay Description:Compound was evaluated for binding affinity against carboxypeptidase A (CPA), expressed as inhibitory constant (Ki)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCarboxypeptidase A1(Bovine)
University of Athens

LigandPNGBDBM50279955(2-Mercaptomethyl-3-p-tolyl-propionic acid | CHEMBL...)
Affinity DataKi:  112nMAssay Description:Binding affinity against carboxypeptidase A using hippurylphenylalanine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCarboxypeptidase A1(Bovine)
University of Athens

LigandPNGBDBM50279955(2-Mercaptomethyl-3-p-tolyl-propionic acid | CHEMBL...)
Affinity DataKi:  112nMAssay Description:Compound was evaluated for binding affinity against carboxypeptidase A (CPA), expressed as inhibitory constant (Ki)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCarboxypeptidase A1(Bovine)
University of Athens

LigandPNGBDBM50279956(2-Mercaptomethyl-3-o-tolyl-propionic acid | CHEMBL...)
Affinity DataKi:  120nMAssay Description:Binding affinity against carboxypeptidase A using hippurylphenylalanine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCarboxypeptidase A1(Bovine)
University of Athens

LigandPNGBDBM50279961(3-(4-Bromo-phenyl)-2-mercaptomethyl-propionic acid...)
Affinity DataKi:  150nMAssay Description:Compound was evaluated for binding affinity against carboxypeptidase A (CPA), expressed as inhibitory constant (Ki)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCarboxypeptidase A1(Bovine)
University of Athens

LigandPNGBDBM50109591(2-Mercaptomethyl-4-methyl-pentanoic acid | CHEMBL3...)
Affinity DataKi:  160nMAssay Description:Inhibition of bovine carboxypeptidase A (CPA) using hippuryl-L-phenylalanine (Hipp-L-Phe) as a substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
University of Athens

LigandPNGBDBM50279963(3-(4-Chloro-phenyl)-2-mercaptomethyl-propionic aci...)
Affinity DataKi:  160nMAssay Description:Compound was evaluated for binding affinity against carboxypeptidase A (CPA), expressed as inhibitory constant (Ki)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCarboxypeptidase A1(Bovine)
University of Athens

LigandPNGBDBM50279953(2-Mercaptomethyl-3-m-tolyl-propionic acid | CHEMBL...)
Affinity DataKi:  170nMAssay Description:Binding affinity against carboxypeptidase A using hippurylphenylalanine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCarboxypeptidase A1(Bovine)
University of Athens

LigandPNGBDBM21472(2-benzyl-3-({1-[2-acetamido-3-(1H-imidazol-4-yl)pr...)
Affinity DataKi:  175nMAssay Description:Continuous assays were performed by recording the fluorescence increase at 405 nm (excitation@ 320 nm) induced by the cleavage of fluorogenic substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2008
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
University of Athens

LigandPNGBDBM50109581((S)2-Benzylamino-3-mercapto-propionic acid | CHEMB...)
Affinity DataKi:  190nMAssay Description:Inhibition of bovine carboxypeptidase A (CPA) using hippuryl-L-phenylalanine (Hipp-L-Phe) as a substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
University of Athens

LigandPNGBDBM50279949(2-Mercaptomethyl-3-naphthalen-2-yl-propionic acid ...)
Affinity DataKi:  200nMAssay Description:Binding affinity against carboxypeptidase A using hippurylphenylalanine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCarboxypeptidase A1(Bovine)
University of Athens

LigandPNGBDBM50365328(CHEMBL1955927)
Affinity DataIC50: 250nMAssay Description:Inhibition of bovine pancreas carboxypeptidase A using N-(4-methoxyphenylazoformyl)-phenylalanine as substrate after 5 mins by colorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
University of Athens

LigandPNGBDBM50279945(3-(3,4-Difluoro-phenyl)-2-mercaptomethyl-propionic...)
Affinity DataKi:  250nMAssay Description:Binding affinity against carboxypeptidase A using hippurylphenylalanine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCarboxypeptidase A1(Bovine)
University of Athens

LigandPNGBDBM50283501(CHEMBL4167456)
Affinity DataIC50: 260nMAssay Description:Inhibition of bovine carboxypeptidase A using N-(4-methoxyphenylazoformyl)-Phe-OH as substrate preincubated for 3 hrs followed by susbtrate addition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2020
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
University of Athens

LigandPNGBDBM50100009(2-(1H-Imidazol-4-yl)-3-phenyl-propionic acid | 2-(...)
Affinity DataKi:  260nMAssay Description:Inhibitory constant of carboxypeptidase A (CPA) in absence of Zinc ion.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
University of Athens

LigandPNGBDBM50109599(2-Benzylamino-3-mercapto-propionic acid | CHEMBL16...)
Affinity DataKi:  270nMAssay Description:Inhibition of bovine carboxypeptidase A (CPA) using hippuryl-L-phenylalanine (Hipp-L-Phe) as a substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
University of Athens

LigandPNGBDBM50279950(3-(2,3-Dimethyl-phenyl)-2-mercaptomethyl-propionic...)
Affinity DataKi:  350nMAssay Description:Binding affinity against carboxypeptidase A using hippurylphenylalanine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCarboxypeptidase A1(Bovine)
University of Athens

LigandPNGBDBM50283541(CHEMBL4176703)
Affinity DataIC50: 470nMAssay Description:Inhibition of bovine carboxypeptidase A using N-(4-methoxyphenylazoformyl)-Phe-OH as substrate preincubated for 3 hrs followed by susbtrate addition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2020
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
University of Athens

LigandPNGBDBM50279957(2-Mercaptomethyl-3-naphthalen-1-yl-propionic acid ...)
Affinity DataKi:  480nMAssay Description:Binding affinity against carboxypeptidase A using hippurylphenylalanine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCarboxypeptidase A1(Bovine)
University of Athens

LigandPNGBDBM50279952(3-(3,4-Dimethyl-phenyl)-2-mercaptomethyl-propionic...)
Affinity DataKi:  492nMAssay Description:Binding affinity against carboxypeptidase A using hippurylphenylalanine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCarboxypeptidase A1(Bovine)
University of Athens

LigandPNGBDBM50121929(2-benzylbutanedioic acid | 2-benzylsuccinic acid |...)
Affinity DataKi:  500nMAssay Description:Inhibition of bovine carboxypeptidase A1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
University of Athens

LigandPNGBDBM50283502(CHEMBL4168849)
Affinity DataIC50: 510nMAssay Description:Inhibition of bovine carboxypeptidase A using N-(4-methoxyphenylazoformyl)-Phe-OH as substrate preincubated for 3 hrs followed by susbtrate addition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2020
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
University of Athens

LigandPNGBDBM50109592((S)2-Isopropylamino-3-mercapto-propionic acid | CH...)
Affinity DataKi:  560nMAssay Description:Inhibition of bovine carboxypeptidase A (CPA) using hippuryl-L-phenylalanine (Hipp-L-Phe) as a substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
University of Athens

LigandPNGBDBM50283507(CHEMBL4163047)
Affinity DataIC50: 570nMAssay Description:Inhibition of bovine carboxypeptidase A using N-(4-methoxyphenylazoformyl)-Phe-OH as substrate preincubated for 3 hrs followed by susbtrate addition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2020
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
University of Athens

LigandPNGBDBM50279946(2-Mercaptomethyl-3-(3,4,5-trifluoro-phenyl)-propio...)
Affinity DataKi:  590nMAssay Description:Binding affinity against carboxypeptidase A using hippurylphenylalanine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCarboxypeptidase A1(Bovine)
University of Athens

LigandPNGBDBM50109589((R)3-Mercapto-2-phenethylamino-propionic acid | CH...)
Affinity DataKi:  610nMAssay Description:Inhibition of bovine carboxypeptidase A (CPA) using hippuryl-L-phenylalanine (Hipp-L-Phe) as a substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
University of Athens

LigandPNGBDBM50121272((2S)-2-[(aminosulfonyl)amino]-3-phenylpropanoic ac...)
Affinity DataKi:  650nMAssay Description:Inhibitory activity against Carboxypeptidase AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
University of Athens

LigandPNGBDBM50277985(CHEMBL4166112)
Affinity DataIC50: 750nMAssay Description:Inhibition of bovine pancreas carboxypeptidase A using N-4-(methoxyphenylazoformyl)-Phe-OH as substrate measured after 5 mins by colorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2020
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
University of Athens

LigandPNGBDBM50109580(3-Mercapto-2-[(naphthalen-1-ylmethyl)-amino]-propi...)
Affinity DataKi:  810nMAssay Description:Inhibition of bovine carboxypeptidase A (CPA) using hippuryl-L-phenylalanine (Hipp-L-Phe) as a substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
University of Athens

LigandPNGBDBM50109601(3-Mercapto-2-(4-methoxy-benzylamino)-propionic aci...)
Affinity DataKi:  850nMAssay Description:Inhibition of bovine carboxypeptidase A (CPA) using hippuryl-L-phenylalanine (Hipp-L-Phe) as a substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
University of Athens

LigandPNGBDBM50283499(CHEMBL4173339)
Affinity DataIC50: 960nMAssay Description:Inhibition of bovine carboxypeptidase A using N-(4-methoxyphenylazoformyl)-Phe-OH as substrate preincubated for 3 hrs followed by susbtrate addition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2020
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
University of Athens

LigandPNGBDBM50283496(CHEMBL4169911)
Affinity DataIC50: 970nMAssay Description:Inhibition of bovine carboxypeptidase A using N-(4-methoxyphenylazoformyl)-Phe-OH as substrate preincubated for 3 hrs followed by susbtrate addition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2020
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
University of Athens

LigandPNGBDBM50283497(CHEMBL4165424)
Affinity DataIC50: 1.04E+3nMAssay Description:Inhibition of bovine carboxypeptidase A using N-(4-methoxyphenylazoformyl)-Phe-OH as substrate preincubated for 3 hrs followed by susbtrate addition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2020
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
University of Athens

LigandPNGBDBM21474(3-({1-[2-acetamido-3-(1H-imidazol-4-yl)propanoyl]p...)
Affinity DataKi:  1.05E+3nMAssay Description:Continuous assays were performed by recording the fluorescence increase at 405 nm (excitation@ 320 nm) induced by the cleavage of fluorogenic substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2008
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
University of Athens

LigandPNGBDBM50109604(2-Isopropylamino-3-mercapto-propionic acid | CHEMB...)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibition of bovine carboxypeptidase A (CPA) using hippuryl-L-phenylalanine (Hipp-L-Phe) as a substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
University of Athens

LigandPNGBDBM50283505(CHEMBL4159372)
Affinity DataIC50: 1.13E+3nMAssay Description:Inhibition of bovine carboxypeptidase A using N-(4-methoxyphenylazoformyl)-Phe-OH as substrate preincubated for 3 hrs followed by susbtrate addition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2020
Entry Details Article
PubMed
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