Compile Data Set for Download or QSAR
Report error Found 133 of affinity data for UniProtKB/TrEMBL: P04191
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50035612(OCTANOIC ACID [3S-[3ALPHA, 3ABETA, 4ALPHA, 6BETA, ...)
Affinity DataKd:  0.200nMAssay Description:Binding affinity to rabbit skeletal muscle SERCA1a preincubated for 5 mins followed by Mg-ATP addition measured over 6 mins by spectrophotometric ana...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2016
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50035612(OCTANOIC ACID [3S-[3ALPHA, 3ABETA, 4ALPHA, 6BETA, ...)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of rabbit sarcoplasmic reticulum calcium ATPase by ATP regeneration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50035612(OCTANOIC ACID [3S-[3ALPHA, 3ABETA, 4ALPHA, 6BETA, ...)
Affinity DataKd:  0.200nMAssay Description:Binding affinity to SERCA1a in sarcoplasmic reticulum vesicles of rabbit skeletal muscle after 2.5 to 6 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50326748((3S,3aR,4S,6S,6aR,7S,8S,9bS)-6-acetoxy-4-(butyrylo...)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of rabbit sarcoplasmic reticulum calcium ATPase by ATP regeneration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50326743((3S,3aR,4S,6S,6aR,7S,8S,9bS)-6-acetoxy-4-(butyrylo...)
Affinity DataKd:  1.5nMAssay Description:Binding affinity to SERCA1a in sarcoplasmic reticulum vesicles of rabbit skeletal muscle after 2.5 to 6 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50326743((3S,3aR,4S,6S,6aR,7S,8S,9bS)-6-acetoxy-4-(butyrylo...)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of rabbit sarcoplasmic reticulum calcium ATPase by ATP regeneration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50431169(CHEMBL2332551)
Affinity DataKd:  1.70nMAssay Description:Binding affinity to SERCA1a in sarcoplasmic reticulum vesicles of rabbit skeletal muscle after 2.5 to 6 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50326738((3S,3aR,4S,6S,6aR,7S,8S,9bS)-4-(butyryloxy)-3,3a-d...)
Affinity DataKd:  2.5nMAssay Description:Binding affinity to SERCA1a in sarcoplasmic reticulum vesicles of rabbit skeletal muscle after 2.5 to 6 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50326737((3S,3aR,4S,6S,6aR,7S,8S,9bS)-3,3a-dihydroxy-3,6,9-...)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of rabbit sarcoplasmic reticulum calcium ATPase by ATP regeneration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50431171(CHEMBL2332104)
Affinity DataKd:  2.60nMAssay Description:Binding affinity to SERCA1a in sarcoplasmic reticulum vesicles of rabbit skeletal muscle after 2.5 to 6 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50326751((3S,3aR,4S,6S,6aR,7S,8S,9bS)-6-acetoxy-4-(butyrylo...)
Affinity DataIC50: 3nMAssay Description:Inhibition of rabbit sarcoplasmic reticulum calcium ATPase by ATP regeneration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50035612(OCTANOIC ACID [3S-[3ALPHA, 3ABETA, 4ALPHA, 6BETA, ...)
Affinity DataIC50: 3.90nMAssay Description:Inhibition of rabbit skeletal muscle SERCA1 assessed as reduction in calcium uptake preincubated for 10 mins followed by ATP addition and measured af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50431174(CHEMBL2332101)
Affinity DataKd:  8.5nMAssay Description:Binding affinity to SERCA1a in sarcoplasmic reticulum vesicles of rabbit skeletal muscle after 2.5 to 6 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50326749((3S,3aR,4S,6S,6aR,7S,8S,9bS)-6-acetoxy-4-(butyrylo...)
Affinity DataIC50: 9nMAssay Description:Inhibition of rabbit sarcoplasmic reticulum calcium ATPase by ATP regeneration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50431170(CHEMBL2332105)
Affinity DataKd:  9.40nMAssay Description:Binding affinity to SERCA1a in sarcoplasmic reticulum vesicles of rabbit skeletal muscle after 2.5 to 6 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50326742((3S,3aR,4S,6S,6aR,7S,8S,9bS)-6-acetoxy-3,3a,4-trih...)
Affinity DataIC50: 10nMAssay Description:Inhibition of rabbit sarcoplasmic reticulum calcium ATPase by ATP regeneration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50326742((3S,3aR,4S,6S,6aR,7S,8S,9bS)-6-acetoxy-3,3a,4-trih...)
Affinity DataKd:  10nMAssay Description:Binding affinity to SERCA1a in sarcoplasmic reticulum vesicles of rabbit skeletal muscle after 2.5 to 6 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50527063(CHEMBL4534285)
Affinity DataKi:  11nMAssay Description:Inhibition of rabbit skeletal muscle microsomes SERCA1aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50431175(CHEMBL2332100)
Affinity DataKd:  11nMAssay Description:Binding affinity to SERCA1a in sarcoplasmic reticulum vesicles of rabbit skeletal muscle after 2.5 to 6 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50326746((3S,3aR,4S,6S,6aR,7S,8S,9bS)-3a-hydroxy-3,6,9-trim...)
Affinity DataIC50: 11.1nMAssay Description:Inhibition of rabbit sarcoplasmic reticulum calcium ATPase by ATP regeneration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50431166(CHEMBL2332554)
Affinity DataKd:  13nMAssay Description:Binding affinity to SERCA1a in sarcoplasmic reticulum vesicles of rabbit skeletal muscle after 2.5 to 6 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50431173(CHEMBL2332102)
Affinity DataKd:  13nMAssay Description:Binding affinity to SERCA1a in sarcoplasmic reticulum vesicles of rabbit skeletal muscle after 2.5 to 6 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50326739((3S,3aR,4S,6S,6aR,7S,8S,9bS)-4-(butyryloxy)-3,3a-d...)
Affinity DataIC50: 15.6nMAssay Description:Inhibition of rabbit sarcoplasmic reticulum calcium ATPase by ATP regeneration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50326738((3S,3aR,4S,6S,6aR,7S,8S,9bS)-4-(butyryloxy)-3,3a-d...)
Affinity DataIC50: 16nMAssay Description:Inhibition of rabbit sarcoplasmic reticulum calcium ATPase by ATP regeneration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50453612(CHEMBL4216774)
Affinity DataKi:  17nMAssay Description:Inhibition of rabbit skeletal muscle microsomes SERCA1aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50615551(CHEMBL5268892)
Affinity DataKi:  18nMAssay Description:Inhibition of SERCA1a in rabbit Sarcoplasmic reticulum assessed as inhibition constant in presence of [gamma-32P]ATP and calcium ionophore A23187 by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50326750((3S,3aR,4S,6S,6aR,7S,8S,9bS)-6-acetoxy-8-(2-(biphe...)
Affinity DataIC50: 18nMAssay Description:Inhibition of rabbit sarcoplasmic reticulum calcium ATPase by ATP regeneration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50527071(CHEMBL4514624)
Affinity DataKi:  18nMAssay Description:Inhibition of rabbit skeletal muscle microsomes SERCA1aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50453611(CHEMBL4207081)
Affinity DataKi:  19nMAssay Description:Inhibition of SERCA1a in rabbit Sarcoplasmic reticulum assessed as inhibition constant in presence of [gamma-32P]ATP and calcium ionophore A23187 by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50453611(CHEMBL4207081)
Affinity DataKi:  19nMAssay Description:Inhibition of rabbit skeletal muscle microsomes SERCA1aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50326745(Octanoic acid(2aS,5aS,7S,7aR,8S,9S,10bS,10cR)-7-bu...)
Affinity DataIC50: 19nMAssay Description:Inhibition of rabbit sarcoplasmic reticulum calcium ATPase by ATP regeneration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50326736((3S,3aR,4S,6S,6aR,7S,8S,9bS)-3,3a,6-trihydroxy-3,6...)
Affinity DataIC50: 20nMAssay Description:Inhibition of rabbit sarcoplasmic reticulum calcium ATPase by ATP regeneration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50431168(CHEMBL2332552)
Affinity DataKd:  20nMAssay Description:Binding affinity to SERCA1a in sarcoplasmic reticulum vesicles of rabbit skeletal muscle after 2.5 to 6 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50326735((3S,3aR,4S,6S,6aR,7S,8S,9bS)-4-(butyryloxy)-3,3a,6...)
Affinity DataIC50: 20nMAssay Description:Inhibition of rabbit sarcoplasmic reticulum calcium ATPase by ATP regeneration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50326741((3S,3aR,4S,6S,6aR,7S,8S,9bS)-6-(2-(biphenyl-4-yl)a...)
Affinity DataIC50: 27nMAssay Description:Inhibition of rabbit sarcoplasmic reticulum calcium ATPase by ATP regeneration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50326752((3S,3aR,4S,6S,6aR,7S,8S,9bS)-6-acetoxy-4-(butyrylo...)
Affinity DataIC50: 44nMAssay Description:Inhibition of rabbit sarcoplasmic reticulum calcium ATPase by ATP regeneration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50431172(CHEMBL2332103)
Affinity DataKd:  55nMAssay Description:Binding affinity to SERCA1a in sarcoplasmic reticulum vesicles of rabbit skeletal muscle after 2.5 to 6 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50326740((3S,3aR,4S,6S,6aR,7S,8S,9bS)-4-(butyryloxy)-3,3a-d...)
Affinity DataIC50: 70nMAssay Description:Inhibition of rabbit sarcoplasmic reticulum calcium ATPase by ATP regeneration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50326753((3S,3aR,4S,6S,6aR,7S,8S,9bS)-6-acetoxy-4-(butyrylo...)
Affinity DataIC50: 70nMAssay Description:Inhibition of rabbit sarcoplasmic reticulum calcium ATPase by ATP regeneration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50326744(Octanoic acid(2aS,5aS,7S,7aR,8S,9S,10bS,10cR)-7,10...)
Affinity DataIC50: 70nMAssay Description:Inhibition of rabbit sarcoplasmic reticulum calcium ATPase by ATP regeneration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50326747((3S,3aR,4S,6S,6aR,7S,8S,9bS)-6-acetoxy-4-(butyrylo...)
Affinity DataIC50: 70nMAssay Description:Inhibition of rabbit sarcoplasmic reticulum calcium ATPase by ATP regeneration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50431167(CHEMBL2332553)
Affinity DataKd:  79nMAssay Description:Binding affinity to SERCA1a in sarcoplasmic reticulum vesicles of rabbit skeletal muscle after 2.5 to 6 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50527068(CHEMBL468766 | CHEBI:17734)
Affinity DataIC50: 90nMAssay Description:Inhibition of rabbit SERCA1b expressed in COS7 cells microsomal membranes preincubated for 10 mins followed by addition of ATP and measured after 40 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50527063(CHEMBL4534285)
Affinity DataIC50: 210nMAssay Description:Inhibition of rabbit SERCA1b expressed in COS7 cells microsomal membranes preincubated for 10 mins followed by addition of ATP and measured after 40 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50527076(CHEMBL4436782)
Affinity DataIC50: 270nMAssay Description:Inhibition of rabbit skeletal muscle microsomes SERCA1aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM34117(hydroquinone derivative, 5a)
Affinity DataIC50: 340nMpH: 7.3 T: 2°CAssay Description:Inhibitory potencies of compounds were determined in a coupled ATPase activity assay using SERCA microsomes at 14 different inhibitor concentrations....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50410532(4-NONYLPHENOL)
Affinity DataIC50: 350nMAssay Description:Inhibition of SERCA1a in rabbit microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50410532(4-NONYLPHENOL)
Affinity DataIC50: 350nMAssay Description:Inhibition of rabbit SERCA1aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50150793(4,4'-(propane-2,2-diyl)bis(2,6-dibromophenol) | 3,...)
Affinity DataIC50: 500nMAssay Description:Inhibition of rabbit skeletal muscle microsomes SERCA1a by enzyme-coupled methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50323389(Calmidazolium | CHEMBL1208858)
Affinity DataIC50: 500nMAssay Description:Inhibition of rabbit skeletal muscle microsomes SERCA1a incubated for 10 mins by enzyme-coupled methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
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